Fragment-based drug discovery

J Med Chem. 2004 Jul 1;47(14):3463-82. doi: 10.1021/jm040031v.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Crystallography, X-Ray
  • Drug Design*
  • Enzyme Inhibitors / chemical synthesis*
  • Enzyme Inhibitors / chemistry*
  • Enzyme Inhibitors / pharmacology
  • Humans
  • Magnetic Resonance Spectroscopy
  • Mass Spectrometry
  • Molecular Weight
  • Protein Binding
  • Structure-Activity Relationship
  • Technology, Pharmaceutical

Substances

  • Enzyme Inhibitors