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Found 112 with Last Name = 'abate' and Initial = 'm'
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036480(2,6-Dichloro-3-(2-morpholin-4-yl-ethoxy)-benzoic a...)
Affinity DataKi:  0.00800nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036476(2,6-Dichloro-3-(4-methyl-piperazine-1-sulfonyl)-be...)
Affinity DataKi:  0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036478(3-Carboxymethoxy-2,6-dichloro-benzoic acid 4-isopr...)
Affinity DataKi:  0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036477(2,6-Dichloro-3-(2-morpholin-4-yl-ethoxy)-benzoic a...)
Affinity DataKi:  0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036481(2,6-Dichloro-3-[(2-dimethylamino-ethyl)-methyl-sul...)
Affinity DataKi:  0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036475(2,6-Dichloro-3-(2-pyrrolidin-1-yl-ethoxy)-benzoic ...)
Affinity DataKi:  0.0140nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036482(2,6-Dichloro-3-(4-methyl-piperazine-1-sulfonyl)-be...)
Affinity DataKi:  0.200nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408224(CHEMBL4164954)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408224(CHEMBL4164954)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408220(CHEMBL4175577)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408226(CHEMBL4167303)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408215(CHEMBL4175177)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408220(CHEMBL4175577)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop

Curated by ChEMBL
LigandPNGBDBM50036479(1,1-Dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulfanylmeth...)
Affinity DataKi:  15nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408226(CHEMBL4167303)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408215(CHEMBL4175177)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408218(CHEMBL4163771)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408222(CHEMBL4174442)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408218(CHEMBL4163771)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408214(CHEMBL4163852)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408219(CHEMBL4165369)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408222(CHEMBL4174442)
Affinity DataKi:  606nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408219(CHEMBL4165369)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408214(CHEMBL4163852)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408227(CHEMBL4171735)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408223(CHEMBL4159313)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408221(CHEMBL4167222)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408217(CHEMBL4173284)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408227(CHEMBL4171735)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408217(CHEMBL4173284)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408221(CHEMBL4167222)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408223(CHEMBL4159313)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408226(CHEMBL4167303)
Affinity DataIC50:  70nMAssay Description:Inhibition of FAAH in human U937 cells using AEA containing [ethanolamine-1-3H]AEA as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoacylglycerol lipase ABHD6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408222(CHEMBL4174442)
Affinity DataIC50:  530nMAssay Description:Inhibition of human ABHD6 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408215(CHEMBL4175177)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of FAAH in human U937 cells using AEA containing [ethanolamine-1-3H]AEA as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidylserine lipase ABHD12(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408224(CHEMBL4164954)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human ABHD12 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408224(CHEMBL4164954)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of FAAH in human U937 cells using AEA containing [ethanolamine-1-3H]AEA as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophosphatidylserine lipase ABHD12(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408226(CHEMBL4167303)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human ABHD12 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoacylglycerol lipase ABHD6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408219(CHEMBL4165369)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ABHD6 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408220(CHEMBL4175577)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of FAAH in human U937 cells using AEA containing [ethanolamine-1-3H]AEA as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoacylglycerol lipase ABHD6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408224(CHEMBL4164954)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ABHD6 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoacylglycerol lipase ABHD6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408226(CHEMBL4167303)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ABHD6 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoacylglycerol lipase ABHD6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408220(CHEMBL4175577)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ABHD6 expressed in HEK293 cells using 2-OG as substrate preincubated for 30 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408218(CHEMBL4163771)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAGL in human U937 cells using 2-OG containing [glycerol-1,2,3-3H]AEA as substrate preincubated for 30 mins followed by substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408223(CHEMBL4159313)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAGL in human U937 cells using 2-OG containing [glycerol-1,2,3-3H]AEA as substrate preincubated for 30 mins followed by substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408217(CHEMBL4173284)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAGL in human U937 cells using 2-OG containing [glycerol-1,2,3-3H]AEA as substrate preincubated for 30 mins followed by substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408219(CHEMBL4165369)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAGL in human U937 cells using 2-OG containing [glycerol-1,2,3-3H]AEA as substrate preincubated for 30 mins followed by substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50408227(CHEMBL4171735)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MAGL in human U937 cells using 2-OG containing [glycerol-1,2,3-3H]AEA as substrate preincubated for 30 mins followed by substrate addit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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