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Found 162 with Last Name = 'abdo' and Initial = 'm'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50017721(1-Methyl-4-(5H-dibenzo(a,d)cycloheptenylidene)pipe...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289603(2-(4-Methyl-piperazin-1-yl)-4,6-di-thiophen-2-yl-p...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289607(4,6-Di-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyri...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289609(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-phenyl-...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289602(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-thiophe...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  10nMAssay Description:Inhibition of human O-GlcNAcase after 5 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289608(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289605(4-Furan-2-yl-6-furan-3-yl-2-(4-methyl-piperazin-1-...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289601(4-Furan-3-yl-6-methyl-2-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289606(2-(4-Methyl-piperazin-1-yl)-4-thiophen-2-yl-pyrimi...)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289601(4-Furan-3-yl-6-methyl-2-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  265nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289605(4-Furan-2-yl-6-furan-3-yl-2-(4-methyl-piperazin-1-...)
Affinity DataKi:  415nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289606(2-(4-Methyl-piperazin-1-yl)-4-thiophen-2-yl-pyrimi...)
Affinity DataKi:  484nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289600(2-(4-Methyl-piperazin-1-yl)-4-phenyl-pyrimidine | ...)
Affinity DataKi:  613nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289607(4,6-Di-furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyri...)
Affinity DataKi:  621nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289608(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327039((3aR,5R,6S,7R,7aR)-5-(Hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  700nMAssay Description:Inhibition of human O-GlcNAcase after 5 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289604(4-Furan-2-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  745nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289604(4-Furan-2-yl-2-(4-methyl-piperazin-1-yl)-pyrimidin...)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289603(2-(4-Methyl-piperazin-1-yl)-4,6-di-thiophen-2-yl-p...)
Affinity DataKi:  972nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289609(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-phenyl-...)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289600(2-(4-Methyl-piperazin-1-yl)-4-phenyl-pyrimidine | ...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]-ketanserin from 5-hydroxytryptamine 2A receptor of rat brain cortexMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289602(4-Furan-3-yl-2-(4-methyl-piperazin-1-yl)-6-thiophe...)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat brain hippocampusMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50406864(CHEMBL4161244)
Affinity DataKi:  6.91E+3nMAssay Description:Non-competitive inhibition of electric eel AChE using varying levels of acetylthiocholine iodide as substrate pretreated for 5 mins followed by subst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267344((S)-3-amino-1-(4-(benzyloxy)phenyl)-4-(1H-imidazol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267344((S)-3-amino-1-(4-(benzyloxy)phenyl)-4-(1H-imidazol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267972((S)-3-Amino-4-(1H-imidazol-4-yl)-1-phenyl-butan-2-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267973((S)-3-amino-1-(4-fluorophenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267974((S)-3-Amino-1-(4-chloro-phenyl)-4-(1H-imidazol-4-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267975((S)-3-Amino-1-(4-bromo-phenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267976((S)-3-Amino-1-biphenyl-4-yl-4-(1H-imidazol-4-yl)-b...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267341((S)-3-amino-4-(1H-imidazol-4-yl)-1-p-tolylbutan-2-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267342((S)-3-Amino-4-(1H-imidazol-4-yl)-1-(4-methoxy-phen...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267343((S)-3-amino-4-(1H-imidazol-4-yl)-1-(4-phenoxypheny...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267345((S)-3-amino-1-(2,4-difluorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267346((S)-3-amino-1-(3,4-dichlorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267371((S)-3-amino-4-(1H-imidazol-4-yl)-1-(perfluoropheny...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267467((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-1-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267468((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-2-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267469((S)-3-amino-1-(benzo[d][1,3]dioxol-5-yl)-4-(1H-imi...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267975((S)-3-Amino-1-(4-bromo-phenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Tehran University Of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50325191((Z)-1-(2-Fluorobenzyl)-4-((6-methoxy-3-oxobenzofur...)
Affinity DataIC50:  10nMAssay Description:Inhibition of electric eel AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267345((S)-3-amino-1-(2,4-difluorophenyl)-4-(1H-imidazol-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM29578(isatin Michael acceptor (IMA) analogue, 13a)
Affinity DataIC50:  12nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267976((S)-3-Amino-1-biphenyl-4-yl-4-(1H-imidazol-4-yl)-b...)
Affinity DataIC50:  12.5nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267468((S)-3-amino-4-(1H-imidazol-4-yl)-1-(naphthalen-2-y...)
Affinity DataIC50:  14.5nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267341((S)-3-amino-4-(1H-imidazol-4-yl)-1-p-tolylbutan-2-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Egyptian National Research Centre

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  15nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267973((S)-3-amino-1-(4-fluorophenyl)-4-(1H-imidazol-4-yl...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidinol dehydrogenase(Brucella suis)
Ecole Nationale Sup£Rieure De Chimie De Montpellier

Curated by ChEMBL
LigandPNGBDBM50267343((S)-3-amino-4-(1H-imidazol-4-yl)-1-(4-phenoxypheny...)
Affinity DataIC50:  16nMAssay Description:Inhibition of Brucella suis histidinol dehydrogenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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