Affinity DataIC50: 1.70nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant
human aromatase (baculovirus/insect cell-expressed) converts the
substrate 7-m...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair