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Found 136 with Last Name = 'abdulla' and Initial = 'mm'
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072313(CHEMBL3408393)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202577(3-[4-(1,2-Dihydro-1,5-dimethyl-2-phenyl-3-oxo-3H-p...)
Affinity DataIC50:  2.30nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089076(CHEMBL3577642)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072316(CHEMBL3408396)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  2.80nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202580(2-Chloro-4-[4-(1,2-dihydro-1,5-dimethyl-2-phenyl-3...)
Affinity DataIC50:  3.30nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202578(3-(1,5-Dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyra...)
Affinity DataIC50:  3.40nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088791(CHEMBL3577634)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202579(2-Hydroxy-4-([4-(1,2-dihydro-1,5-dimethyl-2-phenyl...)
Affinity DataIC50:  3.5nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072315(CHEMBL3408395)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088791(CHEMBL3577634)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202576(1-Phenyl-3-[4-(1,2-Dihydro-1,5-dimethyl-2-phenyl-3...)
Affinity DataIC50:  3.70nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202575(2-[4-(1,2-Dihydro-1,5-dimethyl-2-phenyl-3-oxo-3H-p...)
Affinity DataIC50:  3.90nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202574(2-[4-(1,2-Dihydro-1,5-dimethyl-2-phenyl-3-oxo-3H-p...)
Affinity DataIC50:  4.10nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088855(CHEMBL3577632)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088855(CHEMBL3577632)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088858(CHEMBL3577566)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088896(CHEMBL3577645)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072314(CHEMBL3408394)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202573(4-[4-(1,2-Dihydro-1,5-dimethyl-2-phenyl-3-oxo-3H-p...)
Affinity DataIC50:  4.60nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089083(CHEMBL3577635)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089083(CHEMBL3577635)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089074(CHEMBL3577643)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088857(CHEMBL3577567)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088854(CHEMBL3577633)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202572(6-[4-(1,2-Dihydro-1,5-dimethyl-2-phenyl-3-oxo-3H-p...)
Affinity DataIC50:  5.40nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088854(CHEMBL3577633)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088856(CHEMBL3577631)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of p38alpha MAP kinase (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yueyang Vocational Technical College

LigandPNGBDBM202571(1,2-Dihydro-1,5-dimethyl-2-phenyl-4-thiocyanatoace...)
Affinity DataIC50:  6.70nMpH: 7.5 T: 2°CAssay Description:This fluorescence-based assay measures the rate at which recombinant human aromatase (baculovirus/insect cell-expressed) converts the substrate 7-m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088897(CHEMBL3577644)
Affinity DataIC50:  7nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072312(CHEMBL3408392)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM17054((2S,3R,4R,6R,18R)-18-hydroxy-3-methoxy-2-methyl-4-...)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072281(CHEMBL3408382)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
Cairo University

LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  11nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072310(CHEMBL3408390)
Affinity DataIC50:  12nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072309(CHEMBL3408389)
Affinity DataIC50:  13nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
Cairo University

LigandPNGBDBM167935(1,5-Dimethyl-2-phenyl-4-(6-(phenylsulfonyl)tetrazo...)
Affinity DataIC50:  14nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072308(CHEMBL3408388)
Affinity DataIC50:  14nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
Cairo University

LigandPNGBDBM167938(1',5'-Dimethyl-2'-phenyl-5-(phenylsulf...)
Affinity DataIC50:  15nMT: 2°CAssay Description:A 200-µL reaction system containing DPP-IV (Sigma), a test compound, and 25 mmol/L HEPES buffer (containing 140 mmol/L NaCl, 1% BSA, and 80 mmol/L Mg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072307(CHEMBL3408387)
Affinity DataIC50:  16nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072306(CHEMBL3408386)
Affinity DataIC50:  17nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  18nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072305(CHEMBL3408385)
Affinity DataIC50:  19nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50072304(CHEMBL3408384)
Affinity DataIC50:  20nMAssay Description:Inhibition of CHK1 (unknown origin) using FAM-KKKVSRSGLYRSPSMPENLNRPR-COOH peptide substrate incubated for 1 hr by caliper microfluidic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50088859(CHEMBL3577565)
Affinity DataIC50:  20nMAssay Description:Inhibition of ERK1 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50089077(CHEMBL3577641)
Affinity DataIC50:  21nMAssay Description:Inhibition of ERK2 (unknown origin) using GFP-ATF2 as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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