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Found 15 with Last Name = 'abriel' and Initial = 'h'
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM96504(4-chloranyl-2-(2-naphthalen-1-yloxyethanoylamino)b...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526037(CHEMBL4439848)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526038(CHEMBL4525597)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526034(CHEMBL4540384)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526040(CHEMBL4447880)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526032(CHEMBL4574460)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526035(CHEMBL4472038)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526036(CHEMBL4554529)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526039(CHEMBL4465106)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50350791(LEVOBUPIVACAINE HYDROCHLORIDE)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in CHO cells by whole-cell patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50350791(LEVOBUPIVACAINE HYDROCHLORIDE)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in HEK293 cells assessed as blockade of potassium tail current by whole-cell patch clamp techniqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50350790(BUPIVACAINE HYDROCHLORIDE | Bupivacaine | SAMPL3, ...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in CHO cells by whole-cell patch clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 4(Homo sapiens)
University Of Berne

Curated by ChEMBL
LigandPNGBDBM50526033(CHEBI:28820 | CHEMBL2407182)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of TRPM4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50350790(BUPIVACAINE HYDROCHLORIDE | Bupivacaine | SAMPL3, ...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in HEK293 cells assessed as blockade of potassium tail current by whole-cell patch clamp techniqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50350789(BUPIVACAINE | CHEMBL189827)
Affinity DataIC50:  8.40E+4nMAssay Description:Inhibition of wild-type human ERG channel expressed in HEK293 cells assessed as blockade of potassium tail current by whole-cell patch clamp techniqu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed