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Found 69 with Last Name = 'achilefu' and Initial = 's'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390490(CHEMBL2071603)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390491(CHEMBL2071604)
Affinity DataKi:  0.663nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390492(CHEMBL2071605)
Affinity DataKi:  2.27nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataIC50:  0.200nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390490(CHEMBL2071603)
Affinity DataIC50:  0.281nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130898(CHEMBL408381 | DTPA-Gly(Pip)-Pro-Arg-Gly(PipAm)-Ar...)
Affinity DataIC50:  0.300nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130895(CHEMBL408127 | DTPA-Cha(tr-4-Mam)-Pro-Arg-Gly(PipA...)
Affinity DataIC50:  0.300nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130899(CHEMBL408638 | DTPA-DLys-Pro-Arg-Gly(PipAm)-Arg-Pr...)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130873(CHEMBL409477 | DTPA-Arg-Arg-Pro-Tur-Ile-Leu-OH)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130882(CHEMBL406127 | DTPA-DLys-Pro-Arg-Gly(PipAm)-Arg-Pr...)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130876(CHEMBL404942 | DTPA-DTyr-Glu-Asn-Lys-Pro-Gly(PipAm...)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130885(CHEMBL412699 | DTPA-DLys-Pro-Arg-Phe(4-Gu)-Pro-Tyr...)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130886(CHEMBL437288 | alpha-FITC-Gly(Pip)-Pro-Gly(PipAm)-...)
Affinity DataIC50:  0.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50370236(CHEMBL1790850)
Affinity DataIC50:  0.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130883(CHEMBL406456 | epsilon-FITC-DLys-Pro-Gly(PipAm)-Ar...)
Affinity DataIC50:  0.600nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130875(CHEMBL386387 | DTPA-DTyr-Glu-Asn-Lys-Pro-Gly(PipAm...)
Affinity DataIC50:  0.600nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112639(CHEMBL402688 | pQ-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130888(CHEMBL408534 | alpha-FITC-DLys-Pro-Gly(PipAm)-Arg-...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130896(CHEMBL437707 | DTPA-DTyr-Glu-Asn-Lys-Pro-Gly(PipAm...)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112626(CHEMBL442514 | Carbocyanine derivative)
Affinity DataIC50:  1.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130878(CHEMBL424896 | DTPA-DLys-Pro-Arg-Ala(PipAm)-Arg-Pr...)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112623((FITC-Q-W-A-V-G-H-L-M-NH2) | CHEMBL274327)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130893(CHEMBL439694 | alpha,epsilon-Bis(FITC)-DLys-Pro-Gl...)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390492(CHEMBL2071605)
Affinity DataIC50:  3.52nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50390491(CHEMBL2071604)
Affinity DataIC50:  4.31nMAssay Description:Displacement of [125I]-c(RGDyK) from human integrin alphavbeta3 after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112643((DTPA-P-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2) | CHEMBL442...)
Affinity DataIC50:  4.70nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112611((K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL405669)
Affinity DataIC50:  4.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112640((epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL21696...)
Affinity DataIC50:  4.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112629((epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL38528...)
Affinity DataIC50:  5.70nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112632((alpha-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL428280)
Affinity DataIC50:  5.80nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130890(CHEMBL413192 | DTPA-DLys-Pro-Arg-hAla(PipAm)-Arg-P...)
Affinity DataIC50:  6.30nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112619((G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL408739)
Affinity DataIC50:  7.60nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112633((FITC-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL385928)
Affinity DataIC50:  9.20nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112635((alpha,epsilon-(-FITC)2-K-Q-W-A-V-G-H-L-M-NH2) | C...)
Affinity DataIC50:  9.5nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112620((epsilon-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMB...)
Affinity DataIC50:  9.60nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50370235(CHEMBL1790849)
Affinity DataIC50:  10.2nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112625((K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL269310)
Affinity DataIC50:  10.5nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130887(CHEMBL405160 | DTPA-DLys-ACA-Arg-Gly(PipAm)-Arg-Pr...)
Affinity DataIC50:  11.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130877(CHEMBL407187 | DTPA-DLys-Pro-Gly(PipAm)-Arg-Pro-Ty...)
Affinity DataIC50:  11.9nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112627((alpha-FITC-epsilon-DOTA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112646((alpha-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL4...)
Affinity DataIC50:  15.6nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112614((alpha-FITC-epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50:  20nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112616((alpha,epsilon-(FITC)2-K-G-S-G-Q-W-A-V-G-H-L-M-NH2...)
Affinity DataIC50:  20.5nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130892(CHEMBL405804 | DTPA-DLys-Pro-Gly(PipAm)-Arg-Pro-Ty...)
Affinity DataIC50:  21.7nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50370234(CHEMBL1790851)
Affinity DataIC50:  22.1nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130889(CHEMBL408387 | DTPA-DLys-Pro-Arg-Phe(4-Gu)-Arg-Pro...)
Affinity DataIC50:  24.6nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184908(CHEMBL402661 | cypate-[(RGD)4-NH2]1)
Affinity DataIC50:  25.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin-releasing peptide receptor(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112642((Q-W-A-V-G-H-L-M-NH2) | CHEMBL300318)
Affinity DataIC50:  28.3nMAssay Description:In vitro binding affinity of [111In]-DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184904(CHEMBL206344 | cyclo(RGDfV) (control))
Affinity DataIC50:  28.7nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50130891(CHEMBL413010 | DTPA-DLys-Pro-Gly(PipAm)-Arg-Pro-Ty...)
Affinity DataIC50:  42.4nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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