Compile Data Set for Download or QSAR
maximum 50k data
Found 575 with Last Name = 'agama' and Initial = 'k'
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146559(But-3-enoic acid (R)-1-acetoxymethyl-1-hydroxymeth...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146555(Acetic acid (S)-4-decyloxy-1-hydroxymethyl-3-oxo-1...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146556(Acetic acid (R)-4-decyloxy-1-hydroxymethyl-3-oxo-1...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146558(2,2-Dimethyl-propionic acid (S)-4-dodecyloxy-1-hyd...)
Affinity DataKi:  122nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146554(CHEMBL102042 | Octanoic acid (S)-2-acetoxy-3-hydro...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146557(Acetic acid (R)-4-benzyloxy-1-hydroxymethyl-3-oxo-...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146560(Acetic acid (S)-4-dodecyloxy-1-hydroxymethyl-3-oxo...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50146561(Acetic acid (R)-4-dodecyloxy-1-hydroxymethyl-3-oxo...)
Affinity DataKi:  540nMAssay Description:Binding affinity for protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50388546(CHEMBL213072 | CHEMBL333363)
Affinity DataKi:  3.19E+3nMAssay Description:Competitive inhibition of human recombinant Tdp1 after 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  0.240nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412676(US10399979, Compound 17c)
Affinity DataIC50:  0.890nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412680(US10399979, Compound 17d)
Affinity DataIC50:  1nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412674(US10399979, Compound 17a)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412676(US10399979, Compound 17c)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412687(US10399979, Compound 18)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412675(US10399979, Compound 17b)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412680(US10399979, Compound 17d)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412673(US10399979, Compound 13c)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412674(US10399979, Compound 17a)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412676(US10399979, Compound 17c)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412687(US10399979, Compound 18)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412674(US10399979, Compound 17a)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412687(US10399979, Compound 18)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412690(US10399979, Compound 20a)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412675(US10399979, Compound 17b)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412674(US10399979, Compound 17a)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412687(US10399979, Compound 18)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50466000(CHEMBL4287893)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412676(US10399979, Compound 17c)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412672(US10399979, Compound 13b)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412680(US10399979, Compound 17d)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50466000(CHEMBL4287893)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412671(US10399979, Compound 13a)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412672(US10399979, Compound 13b)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412683(US10399979, Compound 17g)
Affinity DataIC50:  11nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412673(US10399979, Compound 13c)
Affinity DataIC50:  11nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412682(US10399979, Compound 17f)
Affinity DataIC50:  11nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412671(US10399979, Compound 13a)
Affinity DataIC50:  14nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412682(US10399979, Compound 17f)
Affinity DataIC50:  15nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412687(US10399979, Compound 18)
Affinity DataIC50:  15nMAssay Description:Inhibition of JAK3 in human SZ4 cells assessed as reduction in IL2-stimulated STAT5 phosphorylation preincubated for 1 hr followed by IL2 stimulation...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412673(US10399979, Compound 13c)
Affinity DataIC50:  17nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412680(US10399979, Compound 17d)
Affinity DataIC50:  18nMAssay Description:Inhibition of JAK1 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412672(US10399979, Compound 13b)
Affinity DataIC50:  18nMAssay Description:Inhibition of TYK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412672(US10399979, Compound 13b)
Affinity DataIC50:  18nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412682(US10399979, Compound 17f)
Affinity DataIC50:  18nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50466000(CHEMBL4287893)
Affinity DataIC50:  23nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM412689(US10399979, Compound 19b)
Affinity DataIC50:  27nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails ArticlePubMed
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