Compile Data Set for Download or QSAR
maximum 50k data
Found 14 with Last Name = 'ahmadnejad' and Initial = 'm'
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152804((2E)-2-(N-hydroxyimino)-1-(4-methanesulfonylphenyl...)
Affinity DataIC50:  120nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  600nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152806((2E)-2-(4-fluorophenyl)-2-(N-hydroxyimino)-1-(4-me...)
Affinity DataIC50:  1.10E+3nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.10E+3nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  1.85E+4nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152803((2E)-2-(N-hydroxyimino)-1-(4-methanesulfonylphenyl...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152804((2E)-2-(N-hydroxyimino)-1-(4-methanesulfonylphenyl...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152805((2E)-2-(4-chlorophenyl)-2-(N-hydroxyimino)-1-(4-me...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152806((2E)-2-(4-fluorophenyl)-2-(N-hydroxyimino)-1-(4-me...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152803((2E)-2-(N-hydroxyimino)-1-(4-methanesulfonylphenyl...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152805((2E)-2-(4-chlorophenyl)-2-(N-hydroxyimino)-1-(4-me...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152802((2E)-2-(N-hydroxyimino)-1-(4-methanesulfonylphenyl...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Mazandaran University Of Medical Sciences

LigandPNGBDBM152802((2E)-2-(N-hydroxyimino)-1-(4-methanesulfonylphenyl...)
Affinity DataIC50: >1.00E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Mazandaran University Of Medical Sciences

LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.13E+5nMpH: 8.0 T: 2°CAssay Description:Reaction mixtures were prepared in 100 mM Tris澦Cl buffer, pH 8.0 containing 1 然 heme and COX-1 or COX-2 and preincubated for 10 min in a waterbath ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed