Compile Data Set for Download or QSAR
maximum 50k data
Found 16 with Last Name = 'ahmed-belkacem' and Initial = 'a'
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371107(CHEMBL397235)
Affinity DataIC50:  350nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50206310(5-Methoxy-9-oxo-9,10-dihydro-acridine-4-carboxylic...)
Affinity DataIC50:  410nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371104(CHEMBL243167)
Affinity DataIC50:  450nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371110(CHEMBL243168)
Affinity DataIC50:  560nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50370874(CHEMBL221371)
Affinity DataIC50:  700nMAssay Description:Inhibition of BCRP expressed in human HEK293 cells assessed as maximal mitoxantrone accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371108(CHEMBL242513)
Affinity DataIC50:  770nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371114(CHEMBL243169)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50370873(CHEMBL222265)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of BCRP expressed in human HEK293 cells assessed as maximal mitoxantrone accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371109(CHEMBL388886 | GNF-PF-2549)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371106(CHEMBL243813)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371105(CHEMBL243814)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371111(CHEMBL397685)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371112(CHEMBL242943)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM60916(2-hydroxy-10H-acridin-9-one | 2-oxidanyl-10H-acrid...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371113(CHEMBL242512)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371103(CHEMBL242942)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed