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Found 23 with Last Name = 'akamatsu' and Initial = 'y'
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of Flt4 (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)
Affinity DataIC50:  11nMAssay Description:Inhibition of KDR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)
Affinity DataIC50:  18nMAssay Description:Inhibition of GST-Flt1 kinase domain (unknown origin) expressed in baculovirus infected Sf9 cells after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of PDGFR-beta (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)
Affinity DataIC50:  480nMAssay Description:Inhibition of PDGFR-beta (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Flt4 (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of KDR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360804(CHEMBL1934668)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327305(CHEMBL1258849 | N,N-dimethyl-1-(4-(((2-phenyl-2H-1...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327308(CHEMBL1233973 | LAURYL DIMETHYLAMINE-N-OXIDE | N,N...)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of EGFR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of GST-Flt1 kinase domain (unknown origin) expressed in baculovirus infected Sf9 cells after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360803(CHEMBL1934667)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360805(CHEMBL1934669)
Affinity DataIC50:  4.75E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360806(CHEMBL1934670)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327308(CHEMBL1233973 | LAURYL DIMETHYLAMINE-N-OXIDE | N,N...)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360802(CHEMBL1710736)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327304(1-(4-(((1-(4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol...)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327306(CHEMBL1258964 | N-(4-((dimethylamino)methyl)benzyl...)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327307(4-((dimethylamino)methyl)-N-((1-(4-methoxyphenyl)-...)
Affinity DataIC50:  5.88E+4nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute Of Microbial Chemistry (Bikaken)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed