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Found 35 with Last Name = 'akerblom' and Initial = 'e'
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50366760(CHEMBL2369589)
Affinity DataKi:  0.75nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50366760(CHEMBL2369589)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096410(AcAsp-D-Glu-Leu-Glu-Cha-Cys | CHEMBL60967)
Affinity DataKi:  23nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50084685(4-(2-Acetylamino-3-carboxy-propionylamino)-4-(1-{3...)
Affinity DataKi:  25nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096411(AcAsp-Glu-Dif-Ile-Cha-Cys | CHEMBL61390)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50084685(4-(2-Acetylamino-3-carboxy-propionylamino)-4-(1-{3...)
Affinity DataKi:  41nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496205(CHEMBL3125043)
Affinity DataKi:  53nMAssay Description:Inhibition of Hepatitis C virus genotype 1a full length NS3/2K-NS4A protease A156T mutant using Ac-DED(Edans)EEAbupsi[COO]ASK(Dabcyl)-NH2 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096404(AcAsp-Glu-Leu-Glu-Cha-Cys | CHEMBL305570)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496205(CHEMBL3125043)
Affinity DataKi:  110nMAssay Description:Inhibition of Hepatitis C virus genotype 1a full length NS3/2K-NS4A protease D168V mutant using Ac-DED(Edans)EEAbupsi[COO]ASK(Dabcyl)-NH2 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496204(CHEMBL3125169)
Affinity DataKi:  110nMAssay Description:Inhibition of Hepatitis C virus genotype 1a full length NS3/2K-NS4A protease A156T mutant using Ac-DED(Edans)EEAbupsi[COO]ASK(Dabcyl)-NH2 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096405(AcAsp-Glu-Met-Glu-Nal-Cyse | CHEMBL64618)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496204(CHEMBL3125169)
Affinity DataKi:  180nMAssay Description:Inhibition of Hepatitis C virus genotype 1a full length NS3/2K-NS4A protease D168V mutant using Ac-DED(Edans)EEAbupsi[COO]ASK(Dabcyl)-NH2 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096410(AcAsp-D-Glu-Leu-Glu-Cha-Cys | CHEMBL60967)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496205(CHEMBL3125043)
Affinity DataKi:  210nMAssay Description:Inhibition of Hepatitis C virus genotype 1a full length NS3/2K-NS4A protease R155K mutant using Ac-DED(Edans)EEAbupsi[COO]ASK(Dabcyl)-NH2 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096411(AcAsp-Glu-Dif-Ile-Cha-Cys | CHEMBL61390)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096407(AcGlu-Dif-Glu-Cha-Cys | CHEMBL431559)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50084634(4-(2-Acetylamino-3-carboxy-propionylamino)-4-(1-{3...)
Affinity DataKi:  360nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096409(AcAsp-Glu-Met-Glu-Cha-Cys | CHEMBL64867)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096409(AcAsp-Glu-Met-Glu-Cha-Cys | CHEMBL64867)
Affinity DataKi:  440nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096404(AcAsp-Glu-Leu-Glu-Cha-Cys | CHEMBL305570)
Affinity DataKi:  490nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50084634(4-(2-Acetylamino-3-carboxy-propionylamino)-4-(1-{3...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepacivirus C)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50496204(CHEMBL3125169)
Affinity DataKi:  580nMAssay Description:Inhibition of Hepatitis C virus genotype 1a full length NS3/2K-NS4A protease R155K mutant using Ac-DED(Edans)EEAbupsi[COO]ASK(Dabcyl)-NH2 as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096407(AcGlu-Dif-Glu-Cha-Cys | CHEMBL431559)
Affinity DataKi:  700nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096412(AcGlu-Dif-Ile-Cha-Cys | CHEMBL304005)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096405(AcAsp-Glu-Met-Glu-Nal-Cyse | CHEMBL64618)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096401(AcDif-Glu-Cha-Cys | CHEMBL62433)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096412(AcGlu-Dif-Ile-Cha-Cys | CHEMBL304005)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096413(AcAsp-Glu-Dif-Lys-Cha-Cys | CHEMBL294440)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096402(Asp-D-Glu-Leu-Glu-Cha-Cys | CHEMBL303541)
Affinity DataKi:  1.54E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096408(AcDif-Ile-Cha-Cys | CHEMBL293631)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096406(Ac-Glu-Cha-Cys | CHEMBL303340)
Affinity DataKi:  4.10E+3nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096401(AcDif-Glu-Cha-Cys | CHEMBL62433)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096403(AcIle-Cha-Cys | CHEMBL60512)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (full-length)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096408(AcDif-Ile-Cha-Cys | CHEMBL293631)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50096406(Ac-Glu-Cha-Cys | CHEMBL303340)
Affinity DataKi:  2.30E+5nMAssay Description:Inhibitory activity against hepatitis C virus (HCV) NS3 protease (isolated domain)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed