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Found 158 with Last Name = 'albericio' and Initial = 'f'
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088564(CHEMBL3577041)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088560(CHEMBL3577045)
Affinity DataIC50:  18nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088568(CHEMBL3577037)
Affinity DataIC50:  33nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088563(CHEMBL3577042)
Affinity DataIC50:  36nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088565(CHEMBL3577040)
Affinity DataIC50:  36nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088562(CHEMBL3577043)
Affinity DataIC50:  43nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088557(CHEMBL3577048)
Affinity DataIC50:  48nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088559(CHEMBL3577046)
Affinity DataIC50:  49nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM22787(1-acetyl-2,3-dihydro-1H-indole-2,3-dione | Acetyli...)
Affinity DataIC50:  56nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088554(CHEMBL3577036)
Affinity DataIC50:  58nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088561(CHEMBL3577044)
Affinity DataIC50:  60nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088567(CHEMBL3577038)
Affinity DataIC50:  62nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088566(CHEMBL3577039)
Affinity DataIC50:  68nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088555(CHEMBL3577035)
Affinity DataIC50:  72nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50088556(CHEMBL3577034)
Affinity DataIC50:  83nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226429(CHEMBL237354 | [L-arginyl]-N-(2,4-dichlorophenethy...)
Affinity DataIC50:  170nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226436(CHEMBL401228 | [L-arginyl]-[N-(2,4-dichloropheneth...)
Affinity DataIC50:  180nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50246740((4aS,6aS,6bR,8aR,10S,12aR,12bR,14bS)-10-(2-carboxy...)
Affinity DataIC50:  310nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496372(CHEMBL3126478)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226431(CHEMBL237138 | [[N-(2,4-dichlorophenethyl)-N-(6-am...)
Affinity DataIC50:  400nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226430(CHEMBL400008 | [L-arginyl]-[N-[2-(indol-3-yl)ethyl...)
Affinity DataIC50:  520nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50277089(CHEMBL320364 | Oleanolic Acid 3-O-Glutarate)
Affinity DataIC50:  560nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496355(CHEMBL318169)
Affinity DataIC50:  700nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226432(CHEMBL430173 | cis-(L-arginyl)amino-N-(2,4-dichlor...)
Affinity DataIC50:  700nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226435((S)-N-(2,4-dichlorophenethyl)-N-(2-((2,4-dichlorop...)
Affinity DataIC50:  700nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226429(CHEMBL237354 | [L-arginyl]-N-(2,4-dichlorophenethy...)
Affinity DataIC50:  800nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496359(CHEMBL3126474)
Affinity DataIC50:  800nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226434(CHEMBL392540 | [L-arginyl]-N-[2-(indol-3-yl)ethyl]...)
Affinity DataIC50:  1.10E+3nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226433(CHEMBL395124 | [L-arginyl]-[N-[2-(indol-3-yl)-ethy...)
Affinity DataIC50:  1.33E+3nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496357(CHEMBL3126455)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496366(CHEMBL3126468)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496362(CHEMBL3126461)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162761(CHEMBL180302 | [4-Guanidino-1-((S)-4-{(S)-5-[4-((S...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496367(CHEMBL3126466)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162770(CHEMBL180281 | N-[4-Guanidino-1-((S)-4-{(S)-5-[4-(...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226431(CHEMBL237138 | [[N-(2,4-dichlorophenethyl)-N-(6-am...)
Affinity DataIC50:  3.00E+3nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496365(CHEMBL3126454)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50102741(3-O-Acetyloleanolic Acid | Acetyl Oleanolic Acid)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496371(CHEMBL3126467)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496360(CHEMBL3126453)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162764(CHEMBL359680 | [1-((S)-4-{(S)-5-[4-((S)-(S)-2-Benz...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162760(4-Guanidino-N-[(S)-4-((S)-5-{4-[2-(2-imino-imidazo...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162758(4-Guanidino-N-(4-{(S)-5-[4-((S)-4-guanidino-butyry...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidad De Granada

Curated by ChEMBL
LigandPNGBDBM50496361(CHEMBL3126463)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of HIV1 recombinant protease expressed in Escherichia coli using Abz-Ala-Arg-Val-Nle-Tyr(NO2)-Glu-Ala-Nle-NH2 as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162762(CHEMBL181327 | [(S)-4-Guanidino-1-((S)-4-{(S)-5-[4...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162763(CHEMBL181685 | N-((S)-4-{5-[4-(3-Guanidino-propion...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226432(CHEMBL430173 | cis-(L-arginyl)amino-N-(2,4-dichlor...)
Affinity DataIC50:  8.00E+3nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162759(CHEMBL178315 | [1-(4-{(S)-5-[((S)-3-Carbamimidoyl-...)
Affinity DataIC50:  9.09E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50162765((S)-N-[4-Guanidino-1-((S)-4-{(S)-5-[4-(5-guanidino...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibitory concentration against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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