Compile Data Set for Download or QSAR
maximum 50k data
Found 40 with Last Name = 'albiston' and Initial = 'al'
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50331048(CHEMBL1277437 | ethyl 2-acetamido-7-hydroxy-4-(qui...)
Affinity DataKi:  30nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449010(CHEMBL3125960)
Affinity DataKi:  360nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449026(CHEMBL3125936)
Affinity DataKi:  480nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449000(CHEMBL3125942)
Affinity DataKi:  900nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449033(CHEMBL3125949)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449029(CHEMBL3125954)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449011(CHEMBL1604159)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449032(CHEMBL3125950)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449008(CHEMBL3125965)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449007(CHEMBL3125966)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449004(CHEMBL3125937)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449001(CHEMBL3125941)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449030(CHEMBL3125952)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449034(CHEMBL3125948)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50448996(CHEMBL3125931)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50448998(CHEMBL3125944)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449028(CHEMBL3125932)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50448997(CHEMBL3125945)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50448999(CHEMBL1338272)
Affinity DataKi:  7.70E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449027(CHEMBL3125934)
Affinity DataKi:  9.80E+3nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449002(CHEMBL3125940)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449031(CHEMBL3125951)
Affinity DataKi:  1.19E+4nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449003(CHEMBL3125938)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449005(CHEMBL1511289)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449006(CHEMBL3125967)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449009(CHEMBL1303063)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449024(CHEMBL3125961)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449025(CHEMBL1276538)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449014(CHEMBL3125943)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449013(CHEMBL3125935)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449012(CHEMBL1406709)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449023(CHEMBL3125962)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449022(CHEMBL1403937)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449021(CHEMBL1556216)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449020(CHEMBL3125963)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449019(CHEMBL1603587)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449018(CHEMBL3125964)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449015(CHEMBL3125939)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449016(CHEMBL1435420)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Monash Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50449017(CHEMBL1604644)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IRAP in HEKT cells assessed as hydrolysis of L-leucine-4-methyl-7-coumarinylamide after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed