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Found 310 with Last Name = 'ali' and Initial = 'emh'
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50249180(5-((4-(6-chlorothieno[2,3-d]pyrimidin-4-ylamino)pi...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of 5-HT2B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510877(CHEMBL4530036)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510879(CHEMBL4548341)
Affinity DataKi:  524nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510877(CHEMBL4530036)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510875(CHEMBL4447927)
Affinity DataKi:  1.35E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510878(CHEMBL4552737)
Affinity DataKi:  4.06E+3nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510876(CHEMBL4555340)
Affinity DataKi:  5.69E+3nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510878(CHEMBL4552737)
Affinity DataKi:  1.04E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510878(CHEMBL4552737)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510875(CHEMBL4447927)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510877(CHEMBL4530036)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510876(CHEMBL4555340)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510879(CHEMBL4548341)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510879(CHEMBL4548341)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510876(CHEMBL4555340)
Affinity DataKi:  4.08E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)

Curated by ChEMBL
LigandPNGBDBM50510875(CHEMBL4447927)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585092(CHEMBL5087577)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50457446(CHEMBL4212692)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50428286(DABRAFENIB | GSK2118436A)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50428286(DABRAFENIB | GSK2118436A)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585081(CHEMBL5086749)
Affinity DataIC50:  0.980nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM435721(US10570155, Compound 25III | US11332479, Compound ...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585092(CHEMBL5087577)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50560548(CHEMBL4795335)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585085(CHEMBL5080553)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585092(CHEMBL5087577)
Affinity DataIC50:  2nMAssay Description:Inhibition of human wild type BRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585095(CHEMBL5079413)
Affinity DataIC50:  2nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585088(CHEMBL5073246)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585085(CHEMBL5080553)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50563431(CHEMBL4793723)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) using Ser/Thr 03 as substrate after 1 hr in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585088(CHEMBL5073246)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM435721(US10570155, Compound 25III | US11332479, Compound ...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of human wild type BRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585095(CHEMBL5079413)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585093(CHEMBL5092329)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Korea Institute Of Science & Technology (Kist School)

Curated by ChEMBL
LigandPNGBDBM50563437(Arry-614 | Pexmetinib)
Affinity DataIC50:  4nMAssay Description:Inhibition of p38 alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM221688(US10568884, Cpd 9 | US9314464, 9 | US9593100, Comp...)
Affinity DataIC50:  4nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM221688(US10568884, Cpd 9 | US9314464, 9 | US9593100, Comp...)
Affinity DataIC50:  4nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585081(CHEMBL5086749)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human wild type BRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50563432(CHEMBL4797100)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) using Ser/Thr 03 as substrate after 1 hr in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585094(CHEMBL5088891)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585086(CHEMBL5088157)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50560555(CHEMBL4745503)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585096(CHEMBL5076688)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585081(CHEMBL5086749)
Affinity DataIC50:  5nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585097(CHEMBL5079502)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50563427(CHEMBL4758203)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) using Ser/Thr 03 as substrate after 1 hr in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585087(CHEMBL5092112)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585089(CHEMBL5075811)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM435721(US10570155, Compound 25III | US11332479, Compound ...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585085(CHEMBL5080553)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of human wild type BRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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