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Found 39 with Last Name = 'alm' and Initial = 'ra'
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of Helicobacter pylori glutamate racemaseMore data for this Ligand-Target Pair
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215445(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Helicobacter pylori glutamate racemaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215444(5-METHYL-7-(2-METHYLPROPYL)-2-(NAPHTHALEN-1-YLMETH...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Helicobacter pylori glutamate racemaseMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395412(CHEMBL2164745)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395418(CHEMBL2164739)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395395(CHEMBL2163364)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395401(CHEMBL2165061)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395394(CHEMBL2165067)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395413(CHEMBL2164744)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395399(CHEMBL2165063)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395400(CHEMBL2165062)
Affinity DataIC50:  3.90E+4nMAssay Description:Displacement of [3H]-astemizole from human ERG expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395400(CHEMBL2165062)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395393(CHEMBL2165068)
Affinity DataIC50:  5.70E+4nMAssay Description:Displacement of [3H]-astemizole from human ERG expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395419(CHEMBL2165069)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395406(CHEMBL2165056)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395405(CHEMBL2165057)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395402(CHEMBL2165060)
Affinity DataIC50:  9.30E+4nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395409(CHEMBL2164748)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395416(CHEMBL2164741)
Affinity DataIC50:  1.17E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395393(CHEMBL2165068)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395403(CHEMBL2165059)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395410(CHEMBL2164747)
Affinity DataIC50:  1.52E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395417(CHEMBL2164740)
Affinity DataIC50:  1.56E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395396(CHEMBL2165066)
Affinity DataIC50:  1.68E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395411(CHEMBL2164746)
Affinity DataIC50:  1.72E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395408(CHEMBL2165054)
Affinity DataIC50:  1.74E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395404(CHEMBL2165058)
Affinity DataIC50:  1.76E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395407(CHEMBL2165055)
Affinity DataIC50:  1.89E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395397(CHEMBL2165065)
Affinity DataIC50:  1.99E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395397(CHEMBL2165065)
Affinity DataIC50: >2.00E+5nMAssay Description:Displacement of [3H]-astemizole from human ERG expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395398(CHEMBL2165064)
Affinity DataIC50: >2.00E+5nMAssay Description:Displacement of [3H]-astemizole from human ERG expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395398(CHEMBL2165064)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395415(CHEMBL2164742)
Affinity DataIC50:  3.05E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395414(CHEMBL2164743)
Affinity DataIC50: >3.33E+5nMAssay Description:Inhibition of human ERG by Ionworks assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Streptococcus pneumoniae)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215445(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of MurI in Streptococcus pneumoniaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Streptococcus pneumoniae)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215444(5-METHYL-7-(2-METHYLPROPYL)-2-(NAPHTHALEN-1-YLMETH...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of MurI in Streptococcus pneumoniaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215444(5-METHYL-7-(2-METHYLPROPYL)-2-(NAPHTHALEN-1-YLMETH...)
Affinity DataKd:  2.90E+3nMAssay Description:Binding affinity to Helicobacter pylori MurI by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215445(5-(2-((6-chloroquinolin-4-yl)methyl)-7-(cyclopropy...)
Affinity DataKd:  25nMAssay Description:Binding affinity to Helicobacter pylori MurI by protein fluorescence binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
Astrazeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM50215444(5-METHYL-7-(2-METHYLPROPYL)-2-(NAPHTHALEN-1-YLMETH...)
Affinity DataKd:  3.90E+3nMAssay Description:Binding affinity to Helicobacter pylori MurI by protein fluorescence binding assayMore data for this Ligand-Target Pair