Compile Data Set for Download or QSAR
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Found 19 with Last Name = 'amano' and Initial = 'j'
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276373(CHEMBL4125713)
Affinity DataIC50:  800nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276377(CHEMBL4129636)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276378(CHEMBL4126941)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276376(CHEMBL4126909)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276381(CHEMBL4128029)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276381(CHEMBL4128029)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276376(CHEMBL4126909)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276377(CHEMBL4129636)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276372(CHEMBL4128176)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276373(CHEMBL4125713)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276375(CHEMBL4129407)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276372(CHEMBL4128176)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276378(CHEMBL4126941)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276375(CHEMBL4129407)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276380(CHEMBL4127699)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276380(CHEMBL4127699)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276374(CHEMBL4126946)
Affinity DataIC50:  1.60E+6nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Homo sapiens (Human))
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276374(CHEMBL4126946)
Affinity DataIC50:  2.30E+6nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in PMA-differentiated human THP1 cells assessed as reduction in LPS-stimulated IL-1beta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mus musculus)
The Noguchi Institute

Curated by ChEMBL
LigandPNGBDBM50276379(CHEBI:16715 | CHEMBL1234723)
Affinity DataIC50:  2.90E+7nMAssay Description:Inhibition of nigericin-induced NLRP3 inflammasome activation in C57BL/6 mouse bone marrow derived macrophages assessed as reduction in LPS-stimulate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed