Affinity DataKi: 0.600nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of APN in human placenta using AlabetaNA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of APA (unknown origin) using GlubetaNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Competitive inhibition of LAP in porcine kidney microsomesMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of APN in porcine kidney using L-leucine p-nitroanilide as substrate preincubated for 60 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Inhibition of APA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of APN in porcine kidney using Ala-betaNA as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by f...More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition of APA (unknown origin) using GluNA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 870nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of APB in rat testis using ArgbetaNA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.63E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
Affinity DataKi: 2.01E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
Affinity DataKi: 5.95E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
Affinity DataKi: 1.55E+4nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 1.72E+4nMAssay Description:Inhibition of APA (unknown origin) using GlubetaNA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+4nMAssay Description:Inhibition of APA (unknown origin) using GluNA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+4nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Affinity DataKi: 5.60E+4nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 9.00E+4nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <0.170nMAssay Description:Inhibition of HDAC6 (unknown origin) using (FAM)-labeled acetylated peptide as substrate measured after 17 hrs by fluorescence assayMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Inhibition of HDAC6 (unknown origin) using (FAM)-labeled acetylated peptide as substrate measured after 17 hrs by fluorescence assayMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair