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Found 343 with Last Name = 'amin' and Initial = 'sa'
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457465(CHEMBL4204736)
Affinity DataKi:  0.600nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457475(CHEMBL4216408)
Affinity DataKi:  1.5nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  8nMAssay Description:Inhibition of APN in human placenta using AlabetaNA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamyl aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457482(CHEMBL4217064)
Affinity DataKi:  13nMAssay Description:Inhibition of APA (unknown origin) using GlubetaNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457485(CHEMBL4205440)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457467(CHEMBL4217873)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457477(CHEMBL4210855)
Affinity DataKi:  20nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase [435-519](Sus scrofa)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50022748(2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349)
Affinity DataKi:  22nMAssay Description:Competitive inhibition of LAP in porcine kidney microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036969((S)-2-Amino-pentane-1,5-dithiol | CHEMBL101771)
Affinity DataKi:  32nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036827(CHEMBL27040 | [4-(2-Amino-3-mercapto-propyl)-cyclo...)
Affinity DataKi:  35nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  36nMAssay Description:Inhibition of APN in porcine kidney using L-leucine p-nitroanilide as substrate preincubated for 60 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036968((S)-5-Amino-6-mercapto-hexanoic acid hydroxyamide ...)
Affinity DataKi:  37nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataKi:  50nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamyl aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50190112(CHEMBL88808)
Affinity DataKi:  67nMAssay Description:Inhibition of APA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457476(CHEMBL4215801)
Affinity DataKi:  80nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50121710(2-(2,6-Diethyl-phenyl)-4H-isoquinoline-1,3-dione |...)
Affinity DataKi:  120nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457482(CHEMBL4217064)
Affinity DataKi:  120nMAssay Description:Inhibition of APN in porcine kidney using Ala-betaNA as substrate preincubated for 10 mins followed by substrate addition measured after 30 mins by f...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036824((S)-3-Carboxy-1-mercaptomethyl-propyl-ammonium | (...)
Affinity DataKi:  120nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457465(CHEMBL4204736)
Affinity DataKi:  130nMAssay Description:Inhibition of APA (unknown origin) using GluNA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50089194((R)-N*4*-Hydroxy-N*1*-[(S)-1-((S)-2-hydroxymethyl-...)
Affinity DataKi:  170nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036962((S)-4-Carboxy-1-mercaptomethyl-butyl-ammonium | (S...)
Affinity DataKi:  330nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50170890(CHEMBL3806072)
Affinity DataKi:  870nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of APB in rat testis using ArgbetaNA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457484(CHEMBL4206485)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457474(CHEMBL4203613)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457469(CHEMBL4213478)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457463(CHEMBL4073687)
Affinity DataKi:  1.63E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457474(CHEMBL4203613)
Affinity DataKi:  1.95E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457481(CHEMBL4076523)
Affinity DataKi:  2.01E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036818(CHEMBL282364 | [4-(2-Amino-3-mercapto-propyl)-phen...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457481(CHEMBL4076523)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of pig APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457463(CHEMBL4073687)
Affinity DataKi:  5.95E+3nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50036963((R)-4-Carboxy-1-mercaptomethyl-butyl-ammonium | (R...)
Affinity DataKi:  1.55E+4nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  1.72E+4nMAssay Description:Inhibition of APA (unknown origin) using GlubetaNA as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamyl aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457475(CHEMBL4216408)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of APA (unknown origin) using GluNA as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457486(CHEMBL4203901)
Affinity DataKi:  4.50E+4nMAssay Description:Inhibition of hog kidney APN using [3H]Tyr1-Leu5-enkephalin as substrate preincubated for 15 mins followed by substrate addition measured after 15 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457464(CHEMBL4203259)
Affinity DataKi:  5.60E+4nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50457470(CHEMBL4204214)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50526157(CHEMBL4550526)
Affinity DataIC50: <0.170nMAssay Description:Inhibition of HDAC6 (unknown origin) using (FAM)-labeled acetylated peptide as substrate measured after 17 hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206604(CHEMBL3931822)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206615(CHEMBL3903832)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206625(CHEMBL3894894)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206628(CHEMBL3921825)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206607(CHEMBL3960765)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50072082(CHEMBL3407865)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50072077(CHEMBL3407866)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206622(CHEMBL3949189)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Jadavpur University

Curated by ChEMBL
LigandPNGBDBM50526161(CHEMBL4464421)
Affinity DataIC50:  0.790nMAssay Description:Inhibition of HDAC6 (unknown origin) using (FAM)-labeled acetylated peptide as substrate measured after 17 hrs by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206575(CHEMBL3930333)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine 3-monooxygenase(Homo sapiens (Human))
Dr. Hari Singh Gour University

Curated by ChEMBL
LigandPNGBDBM50206630(CHEMBL3922876)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human KMOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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