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Found 179 with Last Name = 'amssoms' and Initial = 'k'
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117542(2-Amino-4-[1-(hydroxycarbamoylmethyl-carbamoyl)-3-...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory constant against amidase free Glutathionylspermidine Synthetase mutant (C79A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118638(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118638(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118640((S)-2-Amino-4-[1-((S)-(S)-2-amino-1-carboxy-ethylc...)
Affinity DataKi:  7.20E+3nMAssay Description:In vitro binding affinity for Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118640((S)-2-Amino-4-[1-((S)-(S)-2-amino-1-carboxy-ethylc...)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118642(5-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118642(5-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118643((S)-2-Amino-4-[1-((S)-(S)-3-amino-1-carboxy-propyl...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118643((S)-2-Amino-4-[1-((S)-(S)-3-amino-1-carboxy-propyl...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118644((S)-2-Amino-4-[1-((S)-(S)-1-carboxy-2-hydroxy-ethy...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118644((S)-2-Amino-4-[1-((S)-(S)-1-carboxy-2-hydroxy-ethy...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118641(6-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118641(6-Amino-2-[(S)-2-((S)-4-amino-4-carboxy-butyrylami...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118639(6-(4-Amino-butylamino)-2-[(S)-2-((S)-4-amino-4-car...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118639(6-(4-Amino-butylamino)-2-[(S)-2-((S)-4-amino-4-car...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118645(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  3.30E+4nMAssay Description:Tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50118645(2-[(S)-2-((S)-4-Amino-4-carboxy-butyrylamino)-4-me...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibitory constant of the compound was tested against glutathionylspermidine synthetase (GspS) in Crithidia fasciculataMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117547(2-Amino-4-[3-methyl-1-(phosphonomethyl-carbamoyl)-...)
Affinity DataKi:  6.00E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition constant of the compound was evaluated against enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathionylspermidine synthase(Crithidia fasciculata)
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50117544(2-amino-4-(1-dihydroxyboronylmethylcarbamoyl-3-met...)
Affinity DataKi:  8.10E+4nMAssay Description:Concentration of the compound required for the inhibition of enzyme Glutathionylspermidine Synthetase wild-type enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50410310(CHEMBL2079773)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243470(US9427440, 18)
Affinity DataIC50:  26nMT: 2°CAssay Description:IC50 con1b were determined according to the method as described previously (Pauwels et al, 2007, J Virol 81:6909-19) using a primer-dependent transcr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243471(US9427440, 19)
Affinity DataIC50:  31nMT: 2°CAssay Description:IC50 con1b were determined according to the method as described previously (Pauwels et al, 2007, J Virol 81:6909-19) using a primer-dependent transcr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243456(US9427440, 1)
Affinity DataIC50:  38nMT: 2°CAssay Description:IC50 con1b were determined according to the method as described previously (Pauwels et al, 2007, J Virol 81:6909-19) using a primer-dependent transcr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243472(US9427440, 20)
Affinity DataIC50:  38nMT: 2°CAssay Description:IC50 con1b were determined according to the method as described previously (Pauwels et al, 2007, J Virol 81:6909-19) using a primer-dependent transcr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243468(US9427440, 16)
Affinity DataIC50:  40nMT: 2°CAssay Description:IC50 con1b were determined according to the method as described previously (Pauwels et al, 2007, J Virol 81:6909-19) using a primer-dependent transcr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50410311(CHEMBL2068731)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422732(CHEMBL424782)
Affinity DataIC50:  112nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422734(CHEMBL368301)
Affinity DataIC50:  178nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422722(CHEMBL360752)
Affinity DataIC50:  186nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (strain HC-J4) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243461(US9427440, 13)
Affinity DataIC50:  190nMpH: 7.5 T: 2°CAssay Description:Measurement of HCV NS5B polymerization activity was performed by evaluating the amount of radiolabeled GTP incorporated by the enzyme in a newly synt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422731(CHEMBL425516)
Affinity DataIC50:  209nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422706(CHEMBL367104)
Affinity DataIC50:  219nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (strain HC-J4) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243457(US9427440, 11)
Affinity DataIC50:  220nMpH: 7.5 T: 2°CAssay Description:Measurement of HCV NS5B polymerization activity was performed by evaluating the amount of radiolabeled GTP incorporated by the enzyme in a newly synt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (strain HC-J4) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243456(US9427440, 1)
Affinity DataIC50:  240nMpH: 7.5 T: 2°CAssay Description:Measurement of HCV NS5B polymerization activity was performed by evaluating the amount of radiolabeled GTP incorporated by the enzyme in a newly synt...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422718(CHEMBL177640)
Affinity DataIC50:  257nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (strain HC-J4) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243460(US9427440, 10)
Affinity DataIC50:  280nMpH: 7.5 T: 2°CAssay Description:Measurement of HCV NS5B polymerization activity was performed by evaluating the amount of radiolabeled GTP incorporated by the enzyme in a newly synt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (strain HC-J4) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243458(US9427440, 5)
Affinity DataIC50:  290nMpH: 7.5 T: 2°CAssay Description:Measurement of HCV NS5B polymerization activity was performed by evaluating the amount of radiolabeled GTP incorporated by the enzyme in a newly synt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422733(CHEMBL414654)
Affinity DataIC50:  355nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422697(CHEMBL362252)
Affinity DataIC50:  372nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422703(CHEMBL366982)
Affinity DataIC50:  380nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (strain HC-J4) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243455(US9427440, 2)
Affinity DataIC50:  410nMpH: 7.5 T: 2°CAssay Description:Measurement of HCV NS5B polymerization activity was performed by evaluating the amount of radiolabeled GTP incorporated by the enzyme in a newly synt...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422699(CHEMBL369841)
Affinity DataIC50:  417nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422711(CHEMBL360274)
Affinity DataIC50:  417nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422700(CHEMBL177515)
Affinity DataIC50:  427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422704(CHEMBL177215)
Affinity DataIC50:  427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422721(CHEMBL177622)
Affinity DataIC50:  427nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422728(CHEMBL424780)
Affinity DataIC50:  437nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Tibotec

Curated by ChEMBL
LigandPNGBDBM50422702(CHEMBL174793)
Affinity DataIC50:  501nMAssay Description:Log of inhibitory concentration against human immunodeficiency virus type 1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein [2420-3010](Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Janssen Ireland

US Patent
LigandPNGBDBM243462(US9427440, 3)
Affinity DataIC50:  530nMT: 2°CAssay Description:IC50 con1b were determined according to the method as described previously (Pauwels et al, 2007, J Virol 81:6909-19) using a primer-dependent transcr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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