TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Umr 8525 Cnrs-Université
Curated by ChEMBL
Umr 8525 Cnrs-Université
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against human glutathione reductaseMore data for this Ligand-Target Pair
TargetGlutathione reductase, mitochondrial(Homo sapiens (Human))
Umr 8525 Cnrs-Université
Curated by ChEMBL
Umr 8525 Cnrs-Université
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibitory concentration against human glutathione reductaseMore data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 4.21E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged human MetAP-1 expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate addition b...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Escherichia coli (strain K12))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 4.55E+4nMAssay Description:Inhibition of C-terminal poly-His-tagged Escherichia coli MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM substrate a...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair