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Found 26 with Last Name = 'andersen' and Initial = 'tl'
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398075(CHEMBL2182012)
Affinity DataKi:  3.50E+3nMAssay Description:Uncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398081(CHEMBL2182013)
Affinity DataKi:  4.00E+3nMAssay Description:Uncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398080(CHEMBL2182014)
Affinity DataKi:  5.00E+3nMAssay Description:Uncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataKi:  1.30E+4nMAssay Description:Noncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataKi:  1.80E+4nMAssay Description:Noncompetitive inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398088(CHEMBL2097001)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of ACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398075(CHEMBL2182012)
Affinity DataIC50:  300nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398076(CHEMBL2182011)
Affinity DataIC50:  300nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398081(CHEMBL2182013)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398075(CHEMBL2182012)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398080(CHEMBL2182014)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398085(CHEMBL2182017)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398086(CHEMBL2182016)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398084(CHEMBL2182020)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398077(CHEMBL1256178)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50:  9.20E+4nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataIC50:  9.90E+4nMAssay Description:Inhibition of plasmin assessed as hydrolysis of H-D-Val-L-Leu-L-Lys-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398078(CHEMBL2182019)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of thrombin assessed as hydrolysis of H-D-Pro-L-Phe-L-Arg-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398079(CHEMBL2182018)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of cathepsin G assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Phe-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398082(CHEMBL2182022)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398087(CHEMBL2182015)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398083(CHEMBL2182021)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human neutrophil elastase assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Val-p-nitroanilide incubated for 2 hrs measured for 20 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398077(CHEMBL1256178)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibition of plasmin assessed as hydrolysis of H-D-Val-L-Leu-L-Lys-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate reader anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50398077(CHEMBL1256178)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of cathepsin G assessed as hydrolysis of N-succinyl-Ala-Ala-Pro-Phe-p-nitroanilide incubated for 2 hrs measured for 20 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed