TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Tested for inhibition of HIV proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Tested for inhibition of HIV proteaseMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:In vitro binding affinity to human luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.331nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 0.851nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards rat Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.37nMAssay Description:Tested for inhibition of HIV proteaseMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:In vitro binding affinity to human luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.97nMAssay Description:Binding affinity towards human Adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Ability to inhibit binding of [3H]-CGS- 21680 to adenosine A2A receptor in rat brain striatal membranes.More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:In vitro binding affinity to human luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of [3H]-CCPA binding to rat adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Binding affinity against human luteinizing releasing hormone receptor cloned in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Ability to inhibit binding of [3H]-CGS- 21680 to adenosine A2A receptor in rat brain striatal membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Ability to inhibit binding of [3H]-CGS- 21680 to adenosine A2A receptor in rat brain striatal membranes.More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:In vitro binding affinity to rat luteinizing hormone-releasing hormone (LHRH) receptor cloned in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair