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Found 389 with Last Name = 'andrei' and Initial = 'g'
TargetAdenosylhomocysteinase(Mus musculus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50006222((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-hydroxymethyl-...)
Affinity DataKi:  3nMAssay Description:Binding affinity of the compound was tested against L929 cells AdoHcy hydrolase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  10nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Mus musculus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50034176(4-(6-Amino-purin-9-yl)-cyclopentane-1,2,3-triol | ...)
Affinity DataKi:  11.1nMAssay Description:Binding affinity of the compound was tested against L929 cells AdoHcy hydrolase activityMore data for this Ligand-Target Pair
TargetAdenosylhomocysteinase(Mus musculus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50008288((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-((R)-1-hydroxy...)
Affinity DataKi:  86nMAssay Description:Inhibitory effect of the compound against L929 Cell S-adenosyl-L-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Mus musculus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50006223(5-(6-Amino-purin-9-yl)-3-methyl-cyclopent-3-ene-1,...)
Affinity DataKi:  150nMAssay Description:Inhibitory effect of the compound against L929 Cell S-adenosyl-L-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490649(CHEMBL2337184)
Affinity DataKi:  260nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490644(CHEMBL2337195)
Affinity DataKi:  310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490643(CHEMBL2337196)
Affinity DataKi:  310nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490669(CHEMBL2337192)
Affinity DataKi:  550nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490662(CHEMBL2337194)
Affinity DataKi:  670nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490668(CHEMBL2337189)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490648(CHEMBL2337186)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490646(CHEMBL2337190)
Affinity DataKi:  1.00E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50369380(CHEMBL606502)
Affinity DataKi:  3.10E+3nMAssay Description:The kinetic constant for inhibition of S-adenosyl-homocysteine hydrolase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50369381(CHEMBL612194)
Affinity DataKi:  3.60E+3nMAssay Description:The kinetic constant for inhibition of S-adenosyl-homocysteine hydrolase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50369379(CHEMBL607755)
Affinity DataKi:  3.90E+3nMAssay Description:The kinetic constant for inhibition of S-adenosyl-homocysteine hydrolase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490660(CHEMBL2337187)
Affinity DataKi:  6.50E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490665(CHEMBL2337181)
Affinity DataKi:  6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490642(CHEMBL2337197)
Affinity DataKi:  6.60E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  7.20E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490659(CHEMBL2337174)
Affinity DataKi:  8.10E+3nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490650(CHEMBL2337183)
Affinity DataKi:  1.00E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490647(CHEMBL2337188)
Affinity DataKi:  1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490645(CHEMBL2337193)
Affinity DataKi:  1.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490653(CHEMBL2337173)
Affinity DataKi:  1.50E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490658(CHEMBL2337175)
Affinity DataKi:  2.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490663(CHEMBL2337191)
Affinity DataKi:  2.90E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490657(CHEMBL2337182)
Affinity DataKi:  4.70E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490652(CHEMBL2337177)
Affinity DataKi:  5.10E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490654(CHEMBL2337201)
Affinity DataKi:  5.20E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Mus musculus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50008289((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-((S)-1-hydroxy...)
Affinity DataKi:  5.57E+4nMAssay Description:Inhibitory effect of the compound against L929 Cell S-adenosyl-L-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490656(CHEMBL2337198)
Affinity DataKi:  6.80E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490661(CHEMBL2337176)
Affinity DataKi:  7.10E+4nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490664(CHEMBL2337185)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490666(CHEMBL2337178)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490667(CHEMBL2337200)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490651(CHEMBL2337179)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490670(CHEMBL2337180)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50490655(CHEMBL2337199)
Affinity DataKi: >1.00E+5nMAssay Description:Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50006222((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-hydroxymethyl-...)
Affinity DataIC50:  7.20nMAssay Description:Tested for inhibitory concentration against S-adenosyl-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50006222((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-hydroxymethyl-...)
Affinity DataIC50:  15.2nMAssay Description:Inhibitory effect against S-adenosyl-L-homocysteine hydrolase of rabbit erythrocyte.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50006222((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-hydroxymethyl-...)
Affinity DataIC50:  15.2nMAssay Description:Inhibitory activity against S-adenosyl-L-homocysteine hydrolase from rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50281613(3-(4-Amino-imidazo[4,5-c]pyridin-1-yl)-5-hydroxyme...)
Affinity DataIC50:  18nMAssay Description:Tested for inhibitory concentration against S-adenosyl-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50281612(5-(4-Amino-imidazo[4,5-c]pyridin-1-yl)-3-hydroxyme...)
Affinity DataIC50:  31nMAssay Description:Tested for inhibitory concentration against S-adenosyl-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50366323((S)-DHPA)
Affinity DataIC50:  280nMAssay Description:Tested for inhibitory concentration against S-adenosyl-homocysteine hydrolaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosylhomocysteinase(Homo sapiens (Human))
Brigham Young University

Curated by ChEMBL
LigandPNGBDBM50008288((1S,2R,5R)-5-(6-Amino-purin-9-yl)-3-((R)-1-hydroxy...)
Affinity DataIC50:  721nMAssay Description:Inhibitory effect against S-adenosyl-L-homocysteine hydrolase of rabbit erythrocyte.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase beta(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50335554(({[({[2-(2-amino-6-oxo-6,9-dihydro-3H-purin-9-yl)e...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human DNA polymerase beta by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA polymerase alpha catalytic subunit(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50335554(({[({[2-(2-amino-6-oxo-6,9-dihydro-3H-purin-9-yl)e...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human DNA polymerase alpha by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 3)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50481118(CHEMBL565370)
Affinity DataIC50:  2.70E+3nMAssay Description:Displacement of [CH3-3H]deoxythymidine from Varicella zoster virus recombinant thymidine kinase after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine kinase(Human herpesvirus 1)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50348873(CHEMBL1807156)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of Herpes simplex virus-1 thymidine kinase-mediated phosphorylation of [methyl-3H]dThd at 1 uM after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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