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Found 128 with Last Name = 'angeli' and Initial = 'l'
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294105(1-(Guanidino)-17-(N1-(methylcyclopropyl)guanidino)...)
Affinity DataKi:  0.0800nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294107(1-(Guanidino)-17-(N1-(beta-methylallyl)guanidino)-...)
Affinity DataKi:  0.5nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294109(1-(Guanidino)-17-(N1-(propargyl)guanidino)-9-azahe...)
Affinity DataKi:  0.700nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294108(1-(Guanidino)-17-(N1-(benzyl)guanidino)-9-azahepta...)
Affinity DataKi:  1nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294106(1-(Guanidino)-17-(N1-(gamma-methylallyl)guanidino)...)
Affinity DataKi:  1.10nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294110(1,1'-(8,8'-azanediylbis(octane-8,1-diyl))bis(3-(3-...)
Affinity DataKi:  1.70nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294104(1-(Guanidino)-17-(N1-(gamma,gamma-dimethylallyl)gu...)
Affinity DataKi:  3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  4nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50032500(1,1'-(8,8'-azanediylbis(octane-8,1-diyl))diguanidi...)
Affinity DataKi:  7.5nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  8nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  9nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294112(1-(5-aminopentyl)-3-(3-methylbut-2-enyl)guanidine ...)
Affinity DataKi:  10nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  10nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294111(1-(4-aminobutyl)-3-(3-methylbut-2-enyl)guanidine |...)
Affinity DataKi:  15nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294113(1-(6-aminohexyl)-3-(3-methylbut-2-enyl)guanidine |...)
Affinity DataKi:  22nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  40nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  65nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294114(1-allyl-3-(4-aminobutyl)guanidine | CHEMBL541766)
Affinity DataKi:  130nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  200nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294095(1-(4-aminobutyl)-3-(prop-2-ynyl)guanidine | CHEMBL...)
Affinity DataKi:  250nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  300nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50129716(1,8-diaminooctane | CHEMBL29392 | OCTANE 1,8-DIAMI...)
Affinity DataKi:  300nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  400nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  500nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  600nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294094(1-(4-aminobutyl)-3-(4-fluorophenyl)guanidine | CHE...)
Affinity DataKi:  630nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294103(4-[N3-gamma,gamma-Dimethyallyl)guanidino]-1-guanid...)
Affinity DataKi:  700nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294100(CHEMBL550832 | N1-(5-Aminopentyl)-N3-(3-methoxyben...)
Affinity DataKi:  1.15E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294102(CHEMBL553638 | N1-[3'-Aminopropyl)-3-aminopropyl]-...)
Affinity DataKi:  1.21E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294096(CHEMBL561237 | N-(3-Methyl-but-2-enyl)-N'-{4-[N'-(...)
Affinity DataKi:  1.50E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294099(CHEMBL561962 | N1-(5-Aminopentyl)-N3[(E)-3-phenyl-...)
Affinity DataKi:  1.53E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294097(CHEMBL550629 | N1-(5-Aminopentyl)-N3-(cyclohexylet...)
Affinity DataKi:  1.72E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294098(CHEMBL552343 | N1-(5-Aminopentyl)-N3-(cyclopropylm...)
Affinity DataKi:  2.58E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM85213(Agmatine | CAS_306-60-5 | CHEMBL58343 | NSC_199 | ...)
Affinity DataKi:  3.00E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine oxidase 1(Zea mays)
Universit£

Curated by ChEMBL
LigandPNGBDBM50294101(CHEMBL558092 | N1-Benzylamine-N3-(gamma,gamma-dime...)
Affinity DataKi:  1.80E+4nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50427868(CHEMBL2326366)
Affinity DataIC50:  16nMAssay Description:Inhibition of MMP-2 (unknown origin) using Mca-Lys-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 as substrate after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50427868(CHEMBL2326366)
Affinity DataIC50:  22nMAssay Description:Inhibition of MMP-13 (unknown origin) using Mca-Lys-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 as substrate after 4 hrs by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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