Affinity DataKi: 0.220nMpH: 7.0Assay Description:The enzyme was assayed at pH 7.0 using the pyruvate kinase/lactate dehydroenase coupling system.More data for this Ligand-Target Pair
Affinity DataKi: 0.470nMpH: 7.0Assay Description:The enzyme was assayed at pH 7.0 using the pyruvate kinase/lactate dehydroenase coupling system.More data for this Ligand-Target Pair
Affinity DataKi: 5nMpH: 7.0Assay Description:The enzyme was assayed at pH 7.0 using the pyruvate kinase/lactate dehydroenase coupling system.More data for this Ligand-Target Pair
Affinity DataKi: 45nMpH: 7.0Assay Description:The enzyme was assayed at pH 7.0 using the pyruvate kinase/lactate dehydroenase coupling system.More data for this Ligand-Target Pair
Affinity DataKi: 140nMpH: 7.0Assay Description:The enzyme was assayed at pH 7.0 using the pyruvate kinase/lactate dehydroenase coupling system.More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
Affinity DataKi: 310nMpH: 7.0Assay Description:The enzyme was assayed at pH 7.0 using the pyruvate kinase/lactate dehydroenase coupling system.More data for this Ligand-Target Pair
Affinity DataKi: 9.60E+5nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+6nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against angiotensin converting enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:The compound was tested for inhibition of purified rat hepatic squalene synthase in the presence of 0.025 mM NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:The compound was tested for inhibition of purified rat hepatic squalene synthase in the presence of 1.2 mM NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibitory activity against angiotensin converting enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+4nMAssay Description:The compound was tested for inhibition of purified rat hepatic squalene synthase in the presence of 0.025 mM NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.23E+5nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+5nMAssay Description:Inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair