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Found 89 with Last Name = 'booker' and Initial = 'g'
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161472(US9108978, 2.02)
Affinity DataKi:  30nM ΔG°:  -44.7kJ/mole IC50:  203nMpH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBifunctional ligase/repressor BirA(Escherichia coli)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  87nMAssay Description:Inhibition of Escherichia coli recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161468(US9108978, 6.09)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/mole IC50:  530nMpH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92383(Biotin triazole, 14)
Affinity DataKi:  90nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388931(CHEMBL2063402)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  182nMAssay Description:Inhibition of human recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388933(CHEMBL2063403)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Escherichia coli)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM161472(US9108978, 2.02)
Affinity DataKi:  225nM ΔG°:  -39.5kJ/molepH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBifunctional ligase/repressor BirA(Escherichia coli)
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM161472(US9108978, 2.02)
Affinity DataKi:  420nM ΔG°:  -37.9kJ/molepH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161470(US9108978, 4.01)
Affinity DataKi:  660nM ΔG°:  -36.7kJ/mole IC50:  4.00E+3nMpH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161469(US9108978, 6.07)
Affinity DataKi:  1.17E+3nM ΔG°:  -35.2kJ/mole IC50:  7.00E+3nMpH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92378(Biotin triazole, 5)
Affinity DataKi:  1.17E+3nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92382(Biotin triazole, 13)
Affinity DataKi:  1.17E+3nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161467(US9108978, 3.25)
Affinity DataKi:  1.83E+3nM ΔG°:  -34.1kJ/mole IC50:  1.16E+4nMpH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388934(CHEMBL2063404)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388927(CHEMBL2063398)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388932(CHEMBL2062535)
Affinity DataKi:  6.43E+3nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM161471(US9108978, 6.34)
Affinity DataKi: >1.00E+4nM ΔG°: >-29.7kJ/mole IC50: >5.00E+4nMpH: 8.0 T: 2°CAssay Description:Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92379(Biotin triazole, 10)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92381(Biotin triazole, 12)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92384(Biotin triazole, 15)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92385(Biotin triazole, 16)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional ligase/repressor BirA(Staphylococcus aureus)
Monash University

US Patent
LigandPNGBDBM92380(Biotin triazole, 11)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro enzyme inhibition using biotin protein ligase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388935(CHEMBL2063405)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201186(CHEMBL3923732)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201187(CHEMBL3976601)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201188(CHEMBL3891635)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201189(CHEMBL3984675)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201190(CHEMBL3942705)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201191(CHEMBL3951442)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201192(CHEMBL3932681)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201193(CHEMBL3974372)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201194(CHEMBL3932600)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201195(CHEMBL3972792)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201196(CHEMBL3961751)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201197(CHEMBL3895686)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201198(CHEMBL3968104)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201199(CHEMBL3934430)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201200(CHEMBL3905875)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201201(CHEMBL3901708)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201202(CHEMBL3971239)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201203(CHEMBL3905724)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201204(CHEMBL3927537)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201205(CHEMBL3914706)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201206(CHEMBL3960176)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201207(CHEMBL3910734)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201208(CHEMBL3892750)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201209(CHEMBL3914868)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50201210(CHEMBL3933745)
Affinity DataKi: >1.60E+4nMAssay Description:Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388928(CHEMBL2063399)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]-biotin from human BPL after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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