TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Abbott Laboratories
Curated by PDSP Ki Database
Abbott Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 5.40E+3nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.15E+4nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.15E+4nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.23E+4nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.30E+4nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of NECA binding to adenosine A2 receptor mediates reduced adenylate cyclase activity in human plateletsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]BH-CCK-8 from Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Virginia School Of Medicine
Curated by ChEMBL
University Of Virginia School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]BH-CCK-8 from Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125I]BH-CCK-8 from Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125I]BH-CCK-8 from Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inhibition of specific binding of [125I]BH-CCK-8 in guinea pig pancreas.More data for this Ligand-Target Pair