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Found 121 with Last Name = 'cutting' and Initial = 'b'
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataKi:  11nMAssay Description:Eq. constant (Ki) for inhibition of Cathepsin K was determined by progress curves, following hydrolysis of Z-Phe-Arg- Amc in the absence and presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113667(4-Benzyloxy-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataKi:  15nMAssay Description:Eq. constant (Ki) for inhibition of Cathepsin K was determined by progress curves, following hydrolysis of Z-Phe-Arg- Amc in the absence and presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347464(CHEMBL1802187)
Affinity DataIC50:  4.80nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113669(1-(2-Chloro-phenyl)-1H-[1,2,4]triazole-3-carboxyli...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113667(4-Benzyloxy-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347465(CHEMBL1802185)
Affinity DataIC50:  6.70nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347449(CHEMBL1171278)
Affinity DataIC50:  10.4nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347450(CHEMBL1802194)
Affinity DataIC50:  11.8nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113674(4-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347451(CHEMBL1802191)
Affinity DataIC50:  15.3nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347452(CHEMBL1802190)
Affinity DataIC50:  16nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347453(CHEMBL1802186)
Affinity DataIC50:  17.1nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347454(CHEMBL1171678)
Affinity DataIC50:  20nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347455(CHEMBL1802188)
Affinity DataIC50:  22nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347456(CHEMBL1802192)
Affinity DataIC50:  23.9nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347457(CHEMBL1802189)
Affinity DataIC50:  27.6nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347458(CHEMBL1802195)
Affinity DataIC50:  29.2nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347459(CHEMBL1802193)
Affinity DataIC50:  38.7nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113673(4-Isopropyl-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataIC50:  65.6nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357403(CHEMBL1917312)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataIC50:  73nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357424(CHEMBL1917473)
Affinity DataIC50:  112nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357407(CHEMBL1917308)
Affinity DataIC50:  135nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357418(CHEMBL1917479)
Affinity DataIC50:  144nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM36025(phenyl-beta-d-glucopyranoside)
Affinity DataIC50:  150nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357423(CHEMBL1917474)
Affinity DataIC50:  153nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357426(CHEMBL1917471)
Affinity DataIC50:  161nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357410(CHEMBL1917305)
Affinity DataIC50:  169nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113665(CHEMBL308392 | [3-Methyl-1-(2-p-tolylamino-ethylca...)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357400(CHEMBL1917484)
Affinity DataIC50:  194nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357422(CHEMBL1917475)
Affinity DataIC50:  196nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357412(CHEMBL1917303)
Affinity DataIC50:  207nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347461(CHEMBL1802183)
Affinity DataIC50:  210nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357417(CHEMBL1917480)
Affinity DataIC50:  216nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357425(CHEMBL1917472)
Affinity DataIC50:  229nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357420(CHEMBL1917477)
Affinity DataIC50:  248nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357421(CHEMBL1917476)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347462(CHEMBL1802184)
Affinity DataIC50:  253nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357411(CHEMBL1917304)
Affinity DataIC50:  296nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357398(CHEMBL1917486)
Affinity DataIC50:  327nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357419(CHEMBL1917478)
Affinity DataIC50:  331nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357399(CHEMBL1917485)
Affinity DataIC50:  333nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357401(CHEMBL1917470)
Affinity DataIC50:  348nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113668(CHEMBL78112 | {1-[2-(4-Chloro-phenylamino)-ethylca...)
Affinity DataIC50:  350nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347463(CHEMBL1170453)
Affinity DataIC50:  364nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357404(CHEMBL1917311)
Affinity DataIC50:  397nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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