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Found 1443 with Last Name = 'ding' and Initial = 'cz'
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339868(4-(1-hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl...)
Affinity DataKi:  20nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339869(5-(1-hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl...)
Affinity DataKi:  20nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339870(2-(1-hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl...)
Affinity DataKi:  80nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339846(6-phenoxybenzo[c][1,2]oxaborol-1(3H)-ol | CHEMBL17...)
Affinity DataKi:  710nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339856(6-(3-methoxyphenoxy)benzo[c][1,2]oxaborol-1(3H)-ol...)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339862(3-(1-hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl...)
Affinity DataKi:  1.44E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339860(6-(3-(benzyloxy)phenoxy)benzo[c][1,2]oxaborol-1(3H...)
Affinity DataKi:  2.27E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339857(6-(3-aminophenoxy)benzo[c][1,2]oxaborol-1(3H)-ol |...)
Affinity DataKi:  2.75E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339859(6-(3-(aminomethyl)phenoxy)benzo[c][1,2]oxaborol-1(...)
Affinity DataKi:  3.33E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339855(6-(phenylamino)benzo[c][1,2]oxaborol-1(3H)-ol | CH...)
Affinity DataKi:  4.73E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280981(2-(3-Chloro-benzyloxy)-ethylamine | CHEMBL65135)
Affinity DataKi:  5.00E+3nMAssay Description:Tested for enzyme affinity with purified bovine liver MAO BMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339867(CHEMBL1761273 | ethyl 4-(1-hydroxy-1,3-dihydrobenz...)
Affinity DataKi:  5.55E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339863(6-(4-methoxyphenoxy)benzo[c][1,2]oxaborol-1(3H)-ol...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339850(6-(hydroxy(phenyl)methyl)benzo[c][1,2]oxaborol-1(3...)
Affinity DataKi:  7.28E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339861(6-(3-((dimethylamino)methyl)phenoxy)benzo[c][1,2]o...)
Affinity DataKi:  7.72E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339858(6-(3-(hydroxymethyl)phenoxy)benzo[c][1,2]oxaborol-...)
Affinity DataKi:  8.40E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339864(6-(4-aminophenoxy)benzo[c][1,2]oxaborol-1(3H)-ol |...)
Affinity DataKi:  8.73E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339847(6-(phenylthio)benzo[c][1,2]oxaborol-1(3H)-ol | CHE...)
Affinity DataKi:  9.09E+3nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339865(6-(4-(aminomethyl)phenoxy)benzo[c][1,2]oxaborol-1(...)
Affinity DataKi:  1.33E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339854(6-((phenylaminooxy)carbonyl)benzo[c][1,2]oxaborol-...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339848(6-benzylbenzo[c][1,2]oxaborol-1(3H)-ol | CHEMBL176...)
Affinity DataKi:  1.98E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339849((1-hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl)(...)
Affinity DataKi:  2.85E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339866(6-(4-((dimethylamino)methyl)phenoxy)benzo[c][1,2]o...)
Affinity DataKi:  4.06E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339853(CHEMBL1761258 | N-(1-hydroxy-1,3-dihydrobenzo[c][1...)
Affinity DataKi:  4.66E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339851(6-(phenylsulfinyl)benzo[c][1,2]oxaborol-1(3H)-ol |...)
Affinity DataKi:  5.80E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Enterobacter cloacae)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50339852(6-(phenylsulfonyl)benzo[c][1,2]oxaborol-1(3H)-ol |...)
Affinity DataKi:  6.32E+4nMAssay Description:Inhibition of Enterobacter cloacae P99 beta-lactamase AmpC P99 using nitrocefin as substrate after 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50042588(5-Aminomethyl-3-[4-(3-chloro-benzyloxy)-phenyl]-ox...)
Affinity DataKi:  6.70E+4nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50042592(3-[4-(3-Chloro-benzyloxy)-phenyl]-5-methylaminomet...)
Affinity DataKi:  2.00E+5nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280981(2-(3-Chloro-benzyloxy)-ethylamine | CHEMBL65135)
Affinity DataKi:  3.40E+5nMAssay Description:Tested for enzyme affinity with purified bovine liver MAO AMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50036731(3-Dimethylamino-1-phenyl-propan-1-one | CHEMBL5011...)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50047897(CHEMBL289199 | Dimethyl-(3-phenyl-propyl)-amine)
Affinity DataKi:  3.80E+5nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50042589(3-[4-(3-Chloro-benzyloxy)-phenyl]-5-dimethylaminom...)
Affinity DataKi:  5.00E+5nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50047898(CHEMBL47794 | Dimethyl-pentyl-amine)
Affinity DataKi:  2.10E+6nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50047896(CHEMBL46232 | Phenethyl-propyl-amine)
Affinity DataKi:  4.00E+6nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50368739(CHEMBL1203212)
Affinity DataKi:  4.70E+6nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50042587(5-Aminomethyl-3-(4-methoxy-phenyl)-dihydro-furan-2...)
Affinity DataKi:  6.70E+6nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50042586(4-Aminomethyl-1-(4-methoxy-phenyl)-pyrrolidin-2-on...)
Affinity DataKi:  6.70E+6nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50018453(CHEMBL46278 | Dimethyl-phenethyl-amine | N,N-dimet...)
Affinity DataKi:  7.10E+6nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016907(CHEMBL46841 | Dimethyl-(4-phenyl-butyl)-amine)
Affinity DataKi:  1.00E+7nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50368566(CHEMBL1203213)
Affinity DataKi:  1.25E+7nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50368737(CHEMBL1203215)
Affinity DataKi:  1.33E+7nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50368741(CHEMBL1203214)
Affinity DataKi:  5.00E+7nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50368738(CHEMBL1203211)
Affinity DataKi:  2.00E+8nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50368740(CHEMBL1203210)
Affinity DataKi:  3.00E+8nMAssay Description:Kinetic constant for inactivation of MAO B from replot of half-lives of inactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM504408(US11040984, Compound 6)
Affinity DataIC50: <0.0150nMAssay Description:Buffer formulation: a buffer consisted of 50 mM HEPES (pH 7.5), 0.01% BSA, 5 mM MgCl2, 0.1 mM Orthovanadate. After the buffer was formulated, an enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM504412(US11040984, Compound 18)
Affinity DataIC50: <0.0150nMAssay Description:Buffer formulation: a buffer consisted of 50 mM HEPES (pH 7.5), 0.01% BSA, 5 mM MgCl2, 0.1 mM Orthovanadate. After the buffer was formulated, an enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM504411(US11040984, Compound 13)
Affinity DataIC50:  0.0160nMAssay Description:Buffer formulation: a buffer consisted of 50 mM HEPES (pH 7.5), 0.01% BSA, 5 mM MgCl2, 0.1 mM Orthovanadate. After the buffer was formulated, an enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM504410(US11040984, Compound 12)
Affinity DataIC50:  0.0170nMAssay Description:Buffer formulation: a buffer consisted of 50 mM HEPES (pH 7.5), 0.01% BSA, 5 mM MgCl2, 0.1 mM Orthovanadate. After the buffer was formulated, an enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor [1-745,751-1210](Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM504403(US11040984, Compound 3)
Affinity DataIC50:  0.0200nMAssay Description:Buffer formulation: a buffer consisted of 50 mM HEPES (pH 7.5), 0.01% BSA, 5 mM MgCl2, 0.1 mM Orthovanadate. After the buffer was formulated, an enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM504415(US11040984, Compound 30)
Affinity DataIC50:  0.0210nMAssay Description:Buffer formulation: a buffer consisted of 50 mM HEPES (pH 7.5), 0.01% BSA, 5 mM MgCl2, 0.1 mM Orthovanadate. After the buffer was formulated, an enzy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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