Affinity DataKi: 6nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of human Thrombin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:The inhibitory activity of the compound was tested against thrombin (IIa)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 70nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of human Thrombin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 200nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of human Thrombin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 300nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of human Thrombin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataKi: 383nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Nv Organon Scientific Development Group
Curated by ChEMBL
Nv Organon Scientific Development Group
Curated by ChEMBL
Affinity DataKi: 675nMAssay Description:The inhibitory activity of the compound was tested against trypsinMore data for this Ligand-Target Pair
TargetSerine protease 1(Bos taurus (bovine))
Nv Organon Scientific Development Group
Curated by ChEMBL
Nv Organon Scientific Development Group
Curated by ChEMBL
Affinity DataKi: 690nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of bovine trypsin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair
Affinity DataKi: 700nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of human Thrombin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:The inhibition constant against human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:The inhibition constant against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
Institute For Biochemistry
Curated by ChEMBL
Institute For Biochemistry
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibitory constant against cAPK (PKA)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of human neutrophil collagenase (Matrix metalloproteinase-8)More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMpH: 7.5Assay Description:Tested for the Inhibition of the catalytic activity of human Thrombin at 25 degree C and pH 7.5.More data for this Ligand-Target Pair