BindingDB PrimarySearch_ki

Found 142 with Last Name = 'mak' and Initial = 'fs'

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

Ki: 1.60nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)

Ki: 5.80nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50176058(2-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-...)

Ki: 6.60nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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Adenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)

Ki: 8.30nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)

Ki: 12nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50176058(2-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-...)

Ki: 72nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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Adenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

Ki: 774nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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Adenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)

Ki: 841nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)

Ki: 2.34E+4nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)

Ki: 4.40E+4nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059885(CHEMBL3394256)

IC50: 18nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059885(CHEMBL3394256)

IC50: 18nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491458(CHEMBL2381774)

IC50: 30nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491458(CHEMBL2381774)

IC50: 30nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059840(CHEMBL3394263)

IC50: 32nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059840(CHEMBL3394263)

IC50: 32nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

IC50: 33nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

IC50: 33nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059796(CHEMBL3394253)

IC50: 35nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059796(CHEMBL3394253)

IC50: 35nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491465(CHEMBL2381773)

IC50: 39nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491465(CHEMBL2381773)

IC50: 39nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059883(CHEMBL3394258)

IC50: 41nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491462(CHEMBL2381761)

IC50: 41nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059883(CHEMBL3394258)

IC50: 41nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491462(CHEMBL2381761)

IC50: 41nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

IC50: 42nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)

IC50: 42nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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3D Structure (crystal)

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491457(CHEMBL2381770)

IC50: 50nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491457(CHEMBL2381770)

IC50: 50nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059799(CHEMBL3394276)

IC50: 59nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059799(CHEMBL3394276)

IC50: 59nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059886(CHEMBL3394255)

IC50: 63nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059886(CHEMBL3394255)

IC50: 63nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059884(CHEMBL3394257)

IC50: 110nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059884(CHEMBL3394257)

IC50: 110nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059848(CHEMBL3394262)

IC50: 120nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059848(CHEMBL3394262)

IC50: 120nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059853(CHEMBL3394261)

IC50: 135nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059853(CHEMBL3394261)

IC50: 135nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491459(CHEMBL2381760)

IC50: 182nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491456(CHEMBL2381757)

IC50: 182nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491459(CHEMBL2381760)

IC50: 182nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50491456(CHEMBL2381757)

IC50: 182nMAssay Description:Antagonist activity at recombinant human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP production after 6...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059872(CHEMBL3394260)

IC50: 437nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059872(CHEMBL3394260)

IC50: 437nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059835(CHEMBL3394265)

IC50: 912nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059835(CHEMBL3394265)

IC50: 912nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

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CHEMBL PC cid PC sid Similars

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059882(CHEMBL3394259)

IC50: 1.07E+3nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL

PNG

BDBM50059882(CHEMBL3394259)

IC50: 1.07E+3nMAssay Description:Inhibition of human adenosine A2A receptor expressed in FlpIn-CHO cells assessed as inhibition of NECA-induced cAMP accumulation incubated for 30 min...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

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