Found 251 with Last Name = 'mustafa' and Initial = 's' 
Affinity DataKi: 0.270nM ΔG°: -50.8kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
3D Structure (crystal)TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 0.270nM ΔG°: -55.5kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 0.540nM ΔG°: -49.2kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor in mouse spleen membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 1.07nM ΔG°: -52.1kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 1.40nM ΔG°: -51.4kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nM ΔG°: -47.0kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity towards alpha-2a adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 1.66nM ΔG°: -51.0kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nM ΔG°: -46.5kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 1.75nM ΔG°: -50.8kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced increase in cAMP accumulation in...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 2.30nM ΔG°: -50.1kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 2.32nM ΔG°: -50.1kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 2.33nM ΔG°: -50.1kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nM ΔG°: -45.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor in rat forebrain membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 2.94nM ΔG°: -49.5kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 3.70nM ΔG°: -48.9kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -44.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 4.70nM ΔG°: -48.3kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 4.77nM ΔG°: -48.3kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
The University Of Tennessee Research Foundation
US Patent
The University Of Tennessee Research Foundation
US Patent
Affinity DataKi: 5.69nM ΔG°: -47.8kJ/moleT: 2°CAssay Description:Cell membranes from HEK293 cells transfected with the human CB1 receptor and membranes from CHO-K1 cells transfected with the human CB2 receptor were...More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nM ΔG°: -43.6kJ/molepH: 7.4 T: 2°CAssay Description:The Ki values were determined by the application of the Cheng-Prusoff equation: Ki = (IC50 x Kd)/(Kd+[L]) where [L] is the concentration of [3H]MIB (...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:In vitro binding affinity towards alpha-2b adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
