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Found 258 with Last Name = 'nicola' and Initial = 'm'
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007887(3-Methyl-2-oxo-2,3-dihydro-benzoimidazole-1-carbox...)
Affinity DataKi:  0.890nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50073179(8-Chloro-11-piperidin-4-ylidene-6,11-dihydro-5H-be...)
Affinity DataKi:  0.970nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000240(CHEMBL435796)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421552(CHEMBL108200)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRelaxin receptor 1(Homo sapiens (Human))
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000252(CHEMBL136347)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000241(CHEMBL138824)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007868(2-Oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid...)
Affinity DataKi:  1.5nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421561(CHEMBL419742)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421562(CHEMBL108889)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000238(CHEMBL336305)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000236(CHEMBL140080)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421567(CHEMBL109937)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007879(3-Methyl-2-oxo-2,3-dihydro-benzoimidazole-1-carbox...)
Affinity DataKi:  1.70nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  1.70nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000255(CHEMBL139088)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000248(CHEMBL139750)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000239(CHEMBL342266)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007884(2-Oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid...)
Affinity DataKi:  2.10nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007870(2-Oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid...)
Affinity DataKi:  2.20nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
Affinity DataKi:  2.30nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000243(CHEMBL423913)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000221(CHEMBL336251)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421554(CHEMBL107875)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000228(CHEMBL136504)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000250(CHEMBL337789)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000242(CHEMBL342443)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000233(CHEMBL136360)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007886(2-Oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid...)
Affinity DataKi:  3.80nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421573(CHEMBL321892)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000254(CHEMBL136213)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421556(CHEMBL109183)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421568(CHEMBL108422)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000253(CHEMBL344847)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007881(4-Methyl-2-oxo-2,3-dihydro-benzoimidazole-1-carbox...)
Affinity DataKi:  7.90nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000220(CHEMBL136709)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421558(CHEMBL432627)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000224(CHEMBL342602)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000245(CHEMBL139150)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50155335(1-{4-[4-(3-{4-[(R)-(4-chlorophenyl)(phenyl)methyl]...)
Affinity DataKi:  9nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000229(CHEMBL139531)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000235(CHEMBL139499)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007858(3-Methyl-2-oxo-2,3-dihydro-benzoimidazole-1-carbox...)
Affinity DataKi:  12nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421553(CHEMBL320535)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM22890(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)
Affinity DataKi:  14nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50155341(1-(4-{4-[3-(4-{13-chloro-4-azatricyclo[9.4.0.0^{3,...)
Affinity DataKi:  14nMAssay Description:Binding affinity towards human histamine H1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Istituto De Angeli

Curated by ChEMBL
LigandPNGBDBM50007882(2-Oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid...)
Affinity DataKi:  16nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000244(CHEMBL140302)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000251(CHEMBL138716)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50000226(CHEMBL139382)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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