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Found 121 with Last Name = 'oleksyszyn' and Initial = 'j'
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244147((4-methoxybenzyl)carbamothioyl(1-aminopentyl)phosp...)
Affinity DataKi:  143nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316047(1-amino-2-methylbutylphosphonic acid monophenylest...)
Affinity DataKi:  230nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)
Affinity DataKi:  230nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316048(1-amino-2-phenylethylphosphonic acid monophenyl es...)
Affinity DataKi:  420nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50024592((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...)
Affinity DataKi:  420nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435121(CHEMBL2391716)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435123(CHEMBL2391713)
Affinity DataKi:  7.80E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435124(CHEMBL2390964)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435117(CHEMBL2391722)
Affinity DataKi:  8.15E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435119(CHEMBL2391719)
Affinity DataKi:  9.40E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435120(CHEMBL2391718)
Affinity DataKi:  9.50E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435116(CHEMBL2391724)
Affinity DataKi:  9.95E+3nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435125(CHEMBL2391726)
Affinity DataKi:  1.11E+4nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435118(CHEMBL2391721)
Affinity DataKi:  1.29E+4nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamyl endopeptidase(Staphylococcus aureus)
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50435122(CHEMBL2391714)
Affinity DataKi:  2.33E+4nMAssay Description:Inhibition of Staphylococcus aureus endoproteinase GluC using Ac-Phe-Leu-Glu-ACC as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316048(1-amino-2-phenylethylphosphonic acid monophenyl es...)
Affinity DataKi:  2.75E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50024592((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...)
Affinity DataKi:  2.75E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316047(1-amino-2-methylbutylphosphonic acid monophenylest...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50129679((1-Amino-3-methyl-butyl)-phosphonic acid | 1-amino...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition of aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184648(CHEMBL378976 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184646(CHEMBL379814 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  53nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184644(CHEMBL377857 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  98nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184647(CHEMBL378778 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  204nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184640(CHEMBL378396 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  208nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204146(1-amino-2-phenylethyl(1-hydroxy-3-phenylpropyl)pho...)
Affinity DataIC50:  240nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184645(CHEMBL209091 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244150((4-methoxybenzyl)carbamothioyl(1-amino-3-phenylpro...)
Affinity DataIC50:  380nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184642(CHEMBL378782 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  455nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244148(1-amino-3-methylbutyl(hexylcarbamothioyl)phosphini...)
Affinity DataIC50:  500nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316042(1-amino-3-phenylpropylphosphonic acid mono-(4-isop...)
Affinity DataIC50:  500nMAssay Description:Inhibition of pig kidney aminopeptidase N using Leu-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204160(1-amino-2-methylpropyl(1-hydroxy-3-phenylpropyl)ph...)
Affinity DataIC50:  500nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204163(CHEMBL227345 | alpha1-(1-amino-3-methylbutane)-alp...)
Affinity DataIC50:  530nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50184643(CHEMBL379807 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  532nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204159(CHEMBL226863 | alpha1-(1-amino-1-phenylmethane)-al...)
Affinity DataIC50:  550nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204161(CHEMBL227290 | bis-alpha-(1-amino-1-phenylmethane)...)
Affinity DataIC50:  600nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244108((4-methoxybenzyl)carbamothioyl(1-aminobutyl)phosph...)
Affinity DataIC50:  680nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204157(CHEMBL227340 | alpha1-(1-amino-1-phenylmethane)-al...)
Affinity DataIC50:  710nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244146(1-aminopentyl(phenethylcarbamothioyl)phosphinic ac...)
Affinity DataIC50:  730nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204149(CHEMBL390323 | bis-alpha-(1-amino-3-phenylpropane)...)
Affinity DataIC50:  830nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204148(CHEMBL227347 | alpha1-(1-amino-2-methylpropane)-al...)
Affinity DataIC50:  930nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
Wroclaw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50204150(1-amino-3-methylbutyl(1-hydroxy-3-phenylpropyl)pho...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316033(1-aminopentylphosphonic acid mono-(4-methylphenyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of pig kidney aminopeptidase N using Leu-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316028(1-aminopropylphosphonic acid mono-(4-tbutylphenyl)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of pig kidney aminopeptidase N using Leu-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244106((4-methoxybenzyl)carbamothioyl(1-aminoethyl)phosph...)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244110(1-amino-2-methylpropyl(hexylcarbamothioyl)phosphin...)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316034(1-aminopentylphosphonic acid mono-(3,4-dimethylphe...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of pig kidney aminopeptidase N using Leu-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50316043(1-amino-3-phenylpropylphosphonic acid mono-(4-t-bu...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of pig kidney aminopeptidase N using Leu-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM50244109(1-amino-2-methylpropyl(isobutylcarbamothioyl)phosp...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of pig kidney aminopeptidase N using Leu-AMC as substrateMore data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
Wroc£?Aw University Of Technology

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of pig kidney aminopeptidase NMore data for this Ligand-Target Pair
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