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Found 49 with Last Name = 'ranganathan' and Initial = 'a'
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKi:  33.9nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKi:  34nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500487(CHEMBL3747370)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]DPCPX from rat cortical membrane adenosine A1 receptor by gamma-scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500487(CHEMBL3747370)
Affinity DataKi:  104nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500487(CHEMBL3747370)
Affinity DataKi:  105nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500492(CHEMBL3746510)
Affinity DataKi:  110nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500492(CHEMBL3746510)
Affinity DataKi:  120nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500490(CHEMBL3747100)
Affinity DataKi:  138nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM68331(N-(1,3-benzothiazol-2-yl)-1-benzothiophene-2-carbo...)
Affinity DataKi:  331nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500490(CHEMBL3747100)
Affinity DataKi:  347nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM89114(MLS-0463381.0001 | N-(5,6-dihydro-4H-cyclopenta[d]...)
Affinity DataKi:  380nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500486(CHEMBL3745825)
Affinity DataKi:  398nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500485(CHEMBL3745803)
Affinity DataKi:  550nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500491(CHEMBL3746858)
Affinity DataKi:  1.82E+3nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500486(CHEMBL3745825)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500489(CHEMBL1417979)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500483(CHEMBL3747257)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500482(CHEMBL1536674)
Affinity DataKi:  2.29E+3nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500493(CHEMBL3746686)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM89114(MLS-0463381.0001 | N-(5,6-dihydro-4H-cyclopenta[d]...)
Affinity DataKi:  2.82E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500487(CHEMBL3747370)
Affinity DataKi:  2.95E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500492(CHEMBL3746510)
Affinity DataKi:  3.09E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500493(CHEMBL3746686)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKi:  3.72E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500494(CHEMBL3746209)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM68331(N-(1,3-benzothiazol-2-yl)-1-benzothiophene-2-carbo...)
Affinity DataKi:  6.17E+3nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500494(CHEMBL3746209)
Affinity DataKi:  1.23E+4nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500488(CHEMBL6215)
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of CA200645 from human adenosine A3 receptor expressed in CHO CRE-SPAP cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500489(CHEMBL1417979)
Affinity DataKi:  2.29E+4nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500483(CHEMBL3747257)
Affinity DataKi:  2.95E+4nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500485(CHEMBL3745803)
Affinity DataKi:  5.62E+4nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500491(CHEMBL3746858)
Affinity DataKi:  6.17E+4nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500488(CHEMBL6215)
Affinity DataKi:  7.59E+4nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500482(CHEMBL1536674)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of CA200645 from human adenosine A1 receptor expressed in CHO cells incubated for 1 hr by fluorescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500485(CHEMBL3745803)
Affinity DataKd:  741nMAssay Description:Competitive antagonist activity at YFP linked human adenosine A3 receptor expressed in CHO CRE-SPAP cells assessed as inhibition of NECA-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
Stockholm University

Curated by ChEMBL
LigandPNGBDBM50500484(CHEMBL3745868)
Affinity DataKd:  741nMAssay Description:Competitive antagonist activity at YFP linked human adenosine A3 receptor expressed in CHO CRE-SPAP cells assessed as inhibition of NECA-induced rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218810(NTS8-13)
Affinity DataKd:  43nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKd:  0.400nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218811(NTSR-H4 inhibitor, 1)
Affinity DataKd:  1.20E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218812(NTSR-H4 inhibitor, 2)
Affinity DataKd:  1.60E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218813(NTSR-H4 inhibitor, 3)
Affinity DataKd:  2.10E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218814(NTSR-H4 inhibitor, 4)
Affinity DataKd:  1.80E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218815(NTSR-H4 inhibitor, 5)
Affinity DataKd:  4.20E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218811(NTSR-H4 inhibitor, 1)
Affinity DataKd:  1.00E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218812(NTSR-H4 inhibitor, 2)
Affinity DataKd:  2.80E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218813(NTSR-H4 inhibitor, 3)
Affinity DataKd:  1.90E+3nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218814(NTSR-H4 inhibitor, 4)
Affinity DataKd:  1.76E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1 [45-272,291-390,C386A,C388A](Rattus norvegicus (Rat))
Stockholm University

LigandPNGBDBM218815(NTSR-H4 inhibitor, 5)
Affinity DataKd:  4.15E+4nMAssay Description:The rat NTSR1 variant NTSR1-H4 was first expressed in E. coli using a derivative of the vector pRG/III-hsMBP. This construct had a C-terminally fused...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed