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Found 2497 with Last Name = 'siu' and Initial = 'm'
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598223((3R,4S)-4-Methyltetrahydrofuran-3-yl(8- amino-6-(8...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598103(US11612606, Compound 452d | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598111(US11612606, Compound 467d | azaspiro[4.4]nonan-3-y...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598119(US11612606, Compound 478b | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598122(US11612606, Compound 479b | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598127((trans)-2-Cyanocyclopentyl(8-amino-7- | US11612606...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598128(US11612606, Compound 482b | fluoro-6-(8-methyl-2,3...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598129((1s,3s)-3-cyanocyclobutyl (8-amino-7- | US11612606...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598130((1s,3s)-3-Cyanocyclobutyl(8-amino-7- | US11612606,...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598132((1s,3s)-3-Hydroxycyclobutyl(8-amino-7- | US1161260...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598133((1r,3r)-3-Hydroxycyclobutyl(8-amino-7- | US1161260...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598134(3-Hydroxy-3-methylcyclobutyl(8-amino- 7-fluoro-6-(...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598136(Cyclobutyl(8-amino-7-fluoro-6-(8- methyl-2,3-dihyd...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598139(2-(2,2-Difluoroethyl)-2- azaspiro[3.3]heptan-6-yl(...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598140((1R,5S,6r)-3-Isopropyl-3- | US11612606, Compound 4...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598141((1R,5S,6r)-3-(oxetan-3-yl)-3- | US11612606, Compou...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598142((R)-6,7-dihydro-5H-pyrrolo[1,2- | US11612606, Comp...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598144((1R,5S,9s)-7-isopropyl-3-oxa-7- | US11612606, Comp...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598145((1R,5S,9s)-7-(2,2-difluoroethyl)-3-oxa-7- | US1161...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598148(1H-pyrido[2,3-b][1,4]oxazin-7- | US11612606, Compo...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598150((R)-8-(Oxetan-3-yl)-8- | US11612606, Compound 511a)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598153((1r,3s)-3-Ethyl-3-hydroxycyclobutyl(8- amino-7-flu...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598155((1r,3r)-3-(1H-Imidazol-1-yl)cyclobutyl | US1161260...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598232((1S,2S)-2-Methylcyclobutyl(8-amino-7- fluoro-6-(8-...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598249((1s,3s)-3-(Hydroxymethyl)cyclobutyl(8- amino-7-flu...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598250((1s,3s)-3-(Methylsulfonyl)cyclobutyl(8- | US116126...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598254((1R,3s)-3-((S)-1- Hydroxyethyl)cyclobutyl(8-amino-...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598256((1s,3s)-3-(2-Hydroxypropan-2- yl)cyclobutyl(8-amin...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598257((1R,5S,9s)-7-(Oxetan-3-yl)-3-oxa-7- | US11612606, ...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598258((1r,3r)-3-Methoxycyclobutyl(8-amino-7- | US1161260...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598260((1r,3r)-3-(Difluoromethyl)cyclobutyl(8- amino-7-fl...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598264(7-Azaspiro[3.5]nonan-2-yl(8-amino-7- fluoro-6-(8-m...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598274(S-(Tetrahydro-2H-pyran-4-yl)(8-amino- 7-fluoro-6-(...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598275(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598276(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598278(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598280(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598282(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598283(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598284(1-(8-Amino-7-fluoro-6-(8-methyl-2,3- dihydro-1H-py...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598285(1-(2-Acetyl-2-azaspiro[3.3]heptan-6-yl)- 3-(8-amin...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598286(1-((3R,4S)-1-Acetyl-3-fluoropiperidin-4-yl)-3-(8-a...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598287((S)-1-(8-Amino-7-fluoro-6-(8-methyl-2,3-dihydro-1H...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598288((R)-1-(8-Amino-7-fluoro-6-(8-methyl- 2,3-dihydro-1...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598289(US11612606, Compound 712ab)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598290(1-(8-Amino-7-fluoro-6-(8-methyl-2,3-dihydro-1H-pyr...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598159((3R,4S)-4-Cyclopropyltetrahydrofuran-3- yl(8-amino...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598160((1s,3s)-3-(Azetidine-1- | US11612606, Compound 517...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598164((1s,3s)-3-(Methylcarbamoyl)cyclobutyl | US11612606...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM598166((1R,5S,6s)-3-(Methylsulfonyl)-3- | US11612606, Com...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 2497 total ) | Next | Last >>
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