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Found 121 with Last Name = 'staab' and Initial = 'a'
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase 12 by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase 2 by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  25nMAssay Description:Inhibition of human carbonic anhydrase 9 by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120038(2-{[2-({6-[1-(1-Carboxy-2-phosphono-ethylcarbamoyl...)
Affinity DataKi:  27nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120023(2-[(2-{[6-(1-Carboxy-2-phosphono-ethylcarbamoyl)-1...)
Affinity DataKi:  73nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120050(2-({2-[6-(1-Carboxy-2-phosphono-ethylcarbamoyl)-1-...)
Affinity DataKi:  100nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120012(2-{[2-(1H-Benzoimidazol-2-ylmethyl)-3-cyclopropylm...)
Affinity DataKi:  140nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120036(2-{[2-(5-Hydroxy-1H-benzoimidazol-2-ylmethyl)-3-me...)
Affinity DataKi:  190nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120027(2-{[3-Methyl-2-(5,6,7-trifluoro-1H-benzoimidazol-2...)
Affinity DataKi:  200nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50103860(2-{[2-(5-Carbamoyl-1H-benzoimidazol-2-ylmethyl)-3-...)
Affinity DataKi:  200nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120048(2-{[2-(5-Methoxy-1H-benzoimidazol-2-ylmethyl)-3-me...)
Affinity DataKi:  200nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120014(2-{[2-(5,6-Difluoro-1H-benzoimidazol-2-ylmethyl)-3...)
Affinity DataKi:  210nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120015(2-({2-[1-(1H-Benzoimidazol-2-yl)-ethyl]-3-methyl-3...)
Affinity DataKi:  230nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120047(2-{[3-Methyl-2-(5-methyl-1H-benzoimidazol-2-ylmeth...)
Affinity DataKi:  240nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120013(2-{[2-(4,6-Difluoro-1H-benzoimidazol-2-ylmethyl)-3...)
Affinity DataKi:  240nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120046(2-({2-[(1H-Benzoimidazol-2-yl)-difluoro-methyl]-3-...)
Affinity DataKi:  250nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  250nMAssay Description:Inhibition of human carbonic anhydrase 1 by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120020(2-{[2-(4,5-Difluoro-1H-benzoimidazol-2-ylmethyl)-3...)
Affinity DataKi:  270nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120033(2-[(2-{Difluoro-[6-(1-methoxycarbonyl-2-phosphono-...)
Affinity DataKi:  277nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120016(2-{[2-(5-Fluoro-1H-benzoimidazol-2-ylmethyl)-3-met...)
Affinity DataKi:  280nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120018(2-{[3-Methyl-2-(4,5,6,7-tetrafluoro-1H-benzoimidaz...)
Affinity DataKi:  280nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120019(2-{[3-Methyl-2-(4,6,7-trifluoro-1H-benzoimidazol-2...)
Affinity DataKi:  350nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120031(2-{[2-(1H-Benzoimidazol-2-ylmethyl)-3-isobutyl-3H-...)
Affinity DataKi:  370nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120035(2-{[2-(5-Chloro-1H-benzoimidazol-2-ylmethyl)-3-met...)
Affinity DataKi:  380nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120034(2-{[3-Methyl-2-(5-trifluoromethyl-1H-benzoimidazol...)
Affinity DataKi:  410nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120051(2-{[2-(1H-Benzoimidazol-2-ylmethyl)-3-methyl-3H-be...)
Affinity DataKi:  450nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120052(2-({2-[(1H-Benzoimidazol-2-yl)-fluoro-methyl]-3-me...)
Affinity DataKi:  470nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120042(2-{[2-(4-Methoxy-1H-benzoimidazol-2-ylmethyl)-3-me...)
Affinity DataKi:  490nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120030(2-({2-[Fluoro-(4,6,7-trifluoro-1H-benzoimidazol-2-...)
Affinity DataKi:  550nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120045(2-{[2-(1H-Benzoimidazol-2-ylmethyl)-3-(2,2-dimethy...)
Affinity DataKi:  610nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120037(2-({2-[(4,6-Difluoro-1H-benzoimidazol-2-yl)-fluoro...)
Affinity DataKi:  660nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120026(2-[2-({2-[(1H-Benzoimidazol-2-yl)-difluoro-methyl]...)
Affinity DataKi:  820nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120028(2-{[2-(1H-Benzoimidazol-2-ylmethyl)-3-(3-methyl-bu...)
Affinity DataKi:  870nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120038(2-{[2-({6-[1-(1-Carboxy-2-phosphono-ethylcarbamoyl...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120046(2-({2-[(1H-Benzoimidazol-2-yl)-difluoro-methyl]-3-...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120049(2-({2-[(6-Carbamoyl-1H-benzoimidazol-2-yl)-difluor...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120041(2-({2-[1-(1H-Benzoimidazol-2-yl)-ethyl]-3-methyl-3...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120010(2-({2-[Difluoro-(5-fluoro-1H-benzoimidazol-2-yl)-m...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120021(2-{[2-(6-Carbamoyl-1H-benzoimidazol-2-ylmethyl)-3-...)
Affinity DataKi:  1.36E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120032(2-({2-[(4,6-Difluoro-1H-benzoimidazol-2-yl)-difluo...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120011(2-({2-[(5-Chloro-1H-benzoimidazol-2-yl)-difluoro-m...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120029(2-({2-[Difluoro-(4,6,7-trifluoro-1H-benzoimidazol-...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120008(2-{[3-Methyl-2-(1-methyl-1H-benzoimidazol-2-ylmeth...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120040(2-({2-[(5,6-Difluoro-1H-benzoimidazol-2-yl)-difluo...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120043(2-{[3-Methyl-2-(4-methyl-1H-benzoimidazol-2-ylmeth...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120029(2-({2-[Difluoro-(4,6,7-trifluoro-1H-benzoimidazol-...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120025(2-{[2-(1H-Benzoimidazol-2-ylmethyl)-3-isopropyl-3H...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of ZnMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120040(2-({2-[(5,6-Difluoro-1H-benzoimidazol-2-yl)-difluo...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120023(2-[(2-{[6-(1-Carboxy-2-phosphono-ethylcarbamoyl)-1...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Celera

Curated by ChEMBL
LigandPNGBDBM50120018(2-{[3-Methyl-2-(4,5,6,7-tetrafluoro-1H-benzoimidaz...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of HCV serine protease NS3/NS4A in the presence of EDTA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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