TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibition of Clostridium botulinum BoNT/A using SNAP-25 (141-206) as substrate by HPLC analysisMore data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincu...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 7.70E+3nMAssay Description:Irreversible inhibition of recombinant Clostridium botulinum N-terminal 6His-tagged BoNT/A (Met1 to Phe425 residues) catalytic domain expressed in Es...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.90E+3nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincu...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.20E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.80E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.10E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.80E+4nMAssay Description:Time dependent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate by me...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 5.20E+4nMAssay Description:Covalent inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincubate...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 6.60E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.80E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincu...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 8.80E+4nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 9.98E+5nMAssay Description:Irreversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide as substrate preincubated...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of Clostridium botulinum BoNT/AMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of 3-HAO in human brain homogenates using [1-14C]-3-HANA as substrate assessed as [14C]-QUIN production after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of 3-HAO in Sprague-Dawley rat brain homogenates using [1-14C]-3-HANA as substrate assessed as [14C]-QUIN production after 1 hr by liquid ...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Reversible inhibition of Clostridium botulinum BoNT/A light chain expressed in Escherichia coli BL21 (DE3) using SNAPtide flp6 as substrate preincuba...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Clostridium botulinum BoNT/A intoxicated in hiPSC-derived neurons assessed as reduction in SNAP-25 cleavage using SNAP-25 as substrate ...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of Clostridium botulinum BoNT/A intoxicated in hiPSC-derived neurons assessed as reduction in SNAP-25 cleavage using SNAP-25 as substrate ...More data for this Ligand-Target Pair
TargetBotulinum neurotoxin type A(Clostridium botulinum)
Boston University School Of Medicine
Curated by ChEMBL
Boston University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of Clostridium botulinum BoNT/A intoxicated in hiPSC-derived neurons assessed as reduction in SNAP-25 cleavage using SNAP-25 as substrate ...More data for this Ligand-Target Pair