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Found 446 with Last Name = 'taylor' and Initial = 'n'
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470598(CHEMBL126050)
Affinity DataKi:  1nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Monash University

Curated by ChEMBL
LigandPNGBDBM50040516(3-(acetylamino)-4-{[amino(iminio)methyl]amino}-2-[...)
Affinity DataKi:  1nMAssay Description:inhibition of Influenza A SialidaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470590(CHEMBL341357)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470604(CHEMBL338825)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470596(CHEMBL125310)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470583(CHEMBL125696)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470587(CHEMBL124648)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  2.5nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from guinea pig tracheaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470605(CHEMBL122169)
Affinity DataKi:  4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470603(CHEMBL124013)
Affinity DataKi:  4nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470582(CHEMBL126043)
Affinity DataKi:  5nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470599(CHEMBL330766)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470595(CHEMBL122019)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.90nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 2 from human expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470592(CHEMBL339311)
Affinity DataKi:  7.90nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470597(CHEMBL330826)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470581(CHEMBL341008)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470606(CHEMBL446099)
Affinity DataKi:  10nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470584(CHEMBL125001)
Affinity DataKi:  13nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470585(CHEMBL415518)
Affinity DataKi:  16nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470607(CHEMBL124624)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470601(CHEMBL123731)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470608(CHEMBL338030)
Affinity DataKi:  20nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Monash University

Curated by ChEMBL
LigandPNGBDBM50040515(3-(acetylamino)-4-ammonio-2-[(1R,2R)-1,2,3-trihydr...)
Affinity DataKi:  40nMAssay Description:inhibition of Influenza A SialidaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92766(PDF inhibitor, compound 8)
Affinity DataKi:  53.7nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470589(CHEMBL331011)
Affinity DataKi:  79nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470594(CHEMBL340405)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470600(CHEMBL435619)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470602(CHEMBL340747)
Affinity DataKi:  100nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92761(PDF inhibitor, compound 3)
Affinity DataKi:  117nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470586(CHEMBL435610)
Affinity DataKi:  126nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470593(CHEMBL126158)
Affinity DataKi:  200nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92764(PDF inhibitor, compound 6)
Affinity DataKi:  213nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92760(PDF inhibitor, compound 2)
Affinity DataKi:  334nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM8885((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...)
Affinity DataKi:  600nMAssay Description:Inhibition of human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataKi:  600nMAssay Description:Inhibitory constant (Ki) for Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92765(PDF inhibitor, compound 7)
Affinity DataKi:  650nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50015985(3-Ethyl-4,5-dihydro-3H-[3,4']bipyridinyl-2,6-dione...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory constant (Ki) for Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470588(CHEMBL340548)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Monash University

Curated by ChEMBL
LigandPNGBDBM50032861(5-((R)-Acetylamino)-4-hydroxy-6-((1R,2R)-1,2,3-tri...)
Affinity DataKi:  4.00E+3nMAssay Description:inhibition of Influenza A SialidaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92759(PDF inhibitor, compound 1)
Affinity DataKi:  6.31E+3nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+3nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from rabbit cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi: <1.00E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from guinea pig tracheaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92762(PDF inhibitor, compound 4)
Affinity DataKi:  2.59E+4nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92763(PDF inhibitor, compound 5)
Affinity DataKi:  3.17E+4nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(GUINEA PIG)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  7.94E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 3 from guinea pig cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Monash University

Curated by ChEMBL
LigandPNGBDBM4942((2R,3R,4S)-4-carbamimidamido-2-(diethylcarbamoyl)-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4942((2R,3R,4S)-4-carbamimidamido-2-(diethylcarbamoyl)-...)
Affinity DataIC50:  1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Monash University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against influenza A virus sialidaseMore data for this Ligand-Target Pair
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