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Found 22 with Last Name = 'thomas' and Initial = 'u'
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11823(Azepane Derivative 4 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  2nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11823(Azepane Derivative 4 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11822((3R,4R)-3-(isonicotinoylamino)azepan-4-yl 4-(2-flu...)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11822((3R,4R)-3-(isonicotinoylamino)azepan-4-yl 4-(2-flu...)
Affinity DataIC50:  5nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11819((3R,4R)-N-{4-[4-(2-hydroxy-5-piperidin-1-ylbenzoyl...)
Affinity DataIC50:  20nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11820((3R,4R)-N-(4-{4-[5-(3,3-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  20nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11817((3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)...)
Affinity DataIC50:  23nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11817((3R,4R)-N-{4-[4-(5-dimethylamino-2-hydroxybenzoyl)...)
Affinity DataIC50:  30nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11824(Azepane Derivative 5 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  39nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11821((3R,4R)-N-(4-{4-[5-(4,4-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  40nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11827(Azepane Derivative 8 | N-((3S,4S)-4-{(E)-2-[4-(2-f...)
Affinity DataIC50:  160nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11824(Azepane Derivative 5 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  355nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11827(Azepane Derivative 8 | N-((3S,4S)-4-{(E)-2-[4-(2-f...)
Affinity DataIC50:  360nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11819((3R,4R)-N-{4-[4-(2-hydroxy-5-piperidin-1-ylbenzoyl...)
Affinity DataIC50:  400nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11818((3R,4R)-N-(4-{4-[3-(3,3-dimethylpiperidin-2-yl)-2-...)
Affinity DataIC50:  750nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11826(Azepane Derivative 7 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  800nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11821((3R,4R)-N-(4-{4-[5-(4,4-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  1.70E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11820((3R,4R)-N-(4-{4-[5-(3,3-dimethylpiperidin-1-yl)-2-...)
Affinity DataIC50:  1.90E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11818((3R,4R)-N-(4-{4-[3-(3,3-dimethylpiperidin-2-yl)-2-...)
Affinity DataIC50:  2.40E+3nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11826(Azepane Derivative 7 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  3.00E+3nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Roche Diagnostics

LigandPNGBDBM11825(Azepane Derivative 6 | N-[(3S,4S)-4-({[4-(2-fluoro...)
Affinity DataIC50:  2.50E+4nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Roche Diagnostics

LigandPNGBDBM11825(Azepane Derivative 6 | N-[(3S,4S)-4-({[4-(2-fluoro...)
Affinity DataIC50:  4.50E+4nMpH: 7.2 T: 2°CAssay Description:In this assay, a fluorescent phosphopeptide tracer and the nonfluorescent phosphopeptides generated during a PKA reaction compete for binding to an a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed