Affinity DataKi: 0.300nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Displacement [3H]LY-186,126 from phosphodiesterase 4 of myocardial vesiclesMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Displacement [3H]LY-186,126 from phosphodiesterase 4 of myocardial vesiclesMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding inhibition against thrombin was measured by nonlinear regression analysis using Morrison's equation for tight-binding inhibitionMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement [3H]LY-186,126 from phosphodiesterase 4 of myocardial vesiclesMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataKi: 6.14E+4nMAssay Description:Displacement [3H]LY-186,126 from phosphodiesterase 4 of myocardial vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of fibrinogen binding to purified Human alphaIIb-beta3 integrin in ELISA with 1% bovine serum albumin (BSA)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Concentration required to reduce binding of fibrinogen to purified Fibrinogen Receptor by 50% using ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of fibrinogen binding to purified human alpha IIb beta3 integrin by 50% in an ELISA testMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of ADP induced platelet aggregation in human platelet-rich plasma (PRP).More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of fibrinogen binding to purified human alpha IIb beta3 integrin by 50% in an ELISA testMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 11.5nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 14.7nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonism of fibrinogen binding to a purified human fibrinogen receptor preparation.More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of fibrinogen binding to purified human alpha IIb beta3 integrin by 50% in an ELISA testMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of ADP induced platelet aggregation in human platelet-rich plasma (PRP).More data for this Ligand-Target Pair
Affinity DataIC50: 24.7nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 28.7nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 31.2nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Concentration required to reduce binding of fibrinogen to purified Fibrinogen Receptor by 50% using ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition ADP-induced (fibrinogen-mediated) platelet aggregation in human platelet-rich plasma (PRP)More data for this Ligand-Target Pair