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Found 120 Enz. Inhib. hit(s) with Target = 'Aldehyde dehydrogenase family 1 member A3'
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50538688(CHEMBL4642789)
Affinity DataKi:  120nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459608(CHEBI:90441 | CHEMBL3276621)
Affinity DataKi:  261nMAssay Description:Inhibition of human ALDH1A3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585949(CHEMBL5083058)
Affinity DataKi:  460nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50527781(CHEMBL4456676)
Affinity DataKi:  540nMAssay Description:Competitive inhibition of recombinant human 6His-tagged ALDH1A3 expressed in Escherichia coli BL21(DE3) using varying level of acetaldehyde as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585950(CHEMBL5075900)
Affinity DataKi: <1.00E+3nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585951(CHEMBL5086460)
Affinity DataKi: <1.00E+3nMAssay Description:Competitive inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as increase in Km without change in Vmax using hexanal as substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataKi:  8.70E+3nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567363(CHEMBL4876602)
Affinity DataIC50:  34nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567386(CHEMBL4861872)
Affinity DataIC50:  50nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567382(CHEMBL4859904)
Affinity DataIC50:  60nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567362(CHEMBL4848258)
Affinity DataIC50:  73nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567372(CHEMBL4875157)
Affinity DataIC50:  89nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459603(CHEMBL4213331)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459603(CHEMBL4213331)
Affinity DataIC50:  90nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567376(CHEMBL4848831)
Affinity DataIC50:  91nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567373(CHEMBL4855442)
Affinity DataIC50:  95nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567374(CHEMBL4849624)
Affinity DataIC50:  100nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567383(CHEMBL4847114)
Affinity DataIC50:  109nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567377(CHEMBL4874309)
Affinity DataIC50:  112nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567366(CHEMBL4876076)
Affinity DataIC50:  119nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459588(CHEMBL4210115)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459588(CHEMBL4210115)
Affinity DataIC50:  120nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567361(CHEMBL4862833)
Affinity DataIC50:  128nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567367(CHEMBL4863668)
Affinity DataIC50:  130nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459613(CHEMBL4214509)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459593(CHEMBL4217452)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567352(CHEMBL4873315)
Affinity DataIC50:  140nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567369(CHEMBL4873090)
Affinity DataIC50:  150nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459602(CHEMBL4216790)
Affinity DataIC50:  170nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459612(CHEMBL4205216)
Affinity DataIC50:  170nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50236905(CHEMBL1349972)
Affinity DataIC50:  170nMAssay Description:Inhibition of full length recombinant human ALDH1A3 expressed in Escherichia coli BL21(DE3) assessed as reduction in dehydrogenase activity by measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567378(CHEMBL4846491)
Affinity DataIC50:  174nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459599(CHEMBL4213859)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567387(CHEMBL4852411)
Affinity DataIC50:  200nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567371(CHEMBL4868666)
Affinity DataIC50:  240nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567385(CHEMBL4846203)
Affinity DataIC50:  250nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585950(CHEMBL5075900)
Affinity DataIC50:  260nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50236900(CHEMBL4072941)
Affinity DataIC50:  270nMAssay Description:In vitro for its ability to displace [3H]- SCH 23390 from Dopamine receptor D1 in bovine striatal membrane expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM69358(3-nitro-4-(1-pyrrolidinyl)benzaldehyde | 3-nitro-4...)
Affinity DataIC50:  270nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585951(CHEMBL5086460)
Affinity DataIC50:  300nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585952(CHEMBL5090970)
Affinity DataIC50:  310nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459586(CHEMBL4217294)
Affinity DataIC50:  390nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50236899(CHEMBL4099822)
Affinity DataIC50:  400nMAssay Description:Inhibition of full length recombinant human ALDH1A3 expressed in Escherichia coli BL21(DE3) assessed as reduction in dehydrogenase activity by measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567384(CHEMBL4849586)
Affinity DataIC50:  480nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567354(CHEMBL4857551)
Affinity DataIC50:  500nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567388(CHEMBL4877915)
Affinity DataIC50:  520nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50585953(CHEMBL5087589)
Affinity DataIC50:  550nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH1A3 assessed as reduction in NADH production using hexanal and NAD+ as substrate by fluori...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50459584(CHEMBL4205099)
Affinity DataIC50:  550nMAssay Description:Inhibition of human recombinant ALDH1A3 assessed as reduction in of NAD(P)H formation incubated for 2 mins by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50572095(CHEMBL4862473)
Affinity DataIC50:  590nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase family 1 member A3(Homo sapiens (Human))
University Of Pisa

Curated by ChEMBL
LigandPNGBDBM50567353(CHEMBL4865571)
Affinity DataIC50:  600nMAssay Description:Inhibition of human ALDH1A3 assessed as NADH formation using propionaldehyde as substrate by spectrophotometeryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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