Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Amphiregulin'
TargetAmphiregulin(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50171860(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)
Affinity DataIC50:  350nMAssay Description:In vitro amphiregulin shedding inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmphiregulin(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50291707((S)-((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquin...)
Affinity DataIC50:  470nMAssay Description:In vitro amphiregulin shedding inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmphiregulin(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50291704((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50:  950nMAssay Description:In vitro amphiregulin shedding inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmphiregulin(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50291705((S)-((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquin...)
Affinity DataIC50:  970nMAssay Description:In vitro amphiregulin shedding inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmphiregulin(Homo sapiens (Human))
Organon K.K.

Curated by ChEMBL
LigandPNGBDBM50291702((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)
Affinity DataIC50:  1.47E+3nMAssay Description:In vitro amphiregulin shedding inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed