Compile Data Set for Download or QSAR
maximum 50k data
Found 921 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3'
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50275902(CHEMBL525577 | D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity to BRS-3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Bag-3 from rat BRS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Bag-3 from rat BRS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86502(CAS_0 | NSC_0 | [D-Tyr6,Beta-Ala11,Phe13,Nle14]Bn(...)
Affinity DataKi:  0.820nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]Bag-3 from mouse BRS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86503(CAS_0 | NSC_0 | [D-Tyr6,Beta-Dap11,Phe13,Nle14]Bn(...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86512(CAS_0 | NSC_0 | [D-Tyr6,(R)-Apa11,Phe13,Nle14]Bn(6...)
Affinity DataKi:  2.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin (6-14) from human BRS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86505(CAS_0 | NSC_0 | [D-Tyr6,(R)-Apa11-4Cl,Phe13,Nle14]...)
Affinity DataKi:  8.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86498(CAS_0 | NSC_0 | [D-Tyr6,(S)-Apa11-3Cl,Phe13,Nle14]...)
Affinity DataKi:  8.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  8.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86509(CAS_0 | NSC_0 | [D-Tyr6,NAlpha-benzoyl-Dap11,Phe13...)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86508(CAS_0 | NSC_0 | [D-Tyr6,NAlpha-acetyl-Dap11,Phe13,...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86498(CAS_0 | NSC_0 | [D-Tyr6,(S)-Apa11-3Cl,Phe13,Nle14]...)
Affinity DataKi:  15.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86504(CAS_0 | NSC_0 | [D-Tyr6,(R)-Apa11-2Cl,Phe13,Nle14]...)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86506(CAS_0 | NSC_0 | [D-Tyr6,(S)-Apa11-2Cl,Phe13,Nle14]...)
Affinity DataKi:  85nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86501(CAS_0 | NSC_0 | [D-Tyr6,(R)-Apa11-3Cl,Phe13,Nle14]...)
Affinity DataKi:  107nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86507(CAS_0 | NSC_0 | [D-Tyr6,Beta-Asp11,Phe13,Nle14]Bn(...)
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86511(CAS_0 | NSC_0 | [D-Tyr6,Beta-Asp(BzlAmd)11,Phe13,N...)
Affinity DataKi:  708nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86510(CAS_0 | NSC_0 | [D-Tyr6,(S)-Apa11-4Cl,Phe13,Nle14]...)
Affinity DataKi:  776nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85495(DPhe6-Bn(6-13)propylamide)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85483(CAS_5748287 | NSC_5748287 | Phyllolitorin)
Affinity DataKi:  2.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85505(Substance P(4-11),[Dpro4,Dtrp7,9,10])
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM86500(CAS_0 | NSC_0 | [D-Tyr6,Beta-Ala11,Phe13,Beta-Dap(...)
Affinity DataKi:  2.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50063814(CHEMBL217438 | Dnal,Cys,Tyr,DTrp,Lys,Val,Cys,Nal-n...)
Affinity DataKi:  2.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85506(CAS_125988 | NSC_125988 | Rhodei-Litorin)
Affinity DataKi:  3.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85482(DPhe6-Bn(6-13)hexylamide)
Affinity DataKi:  3.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85497(Alytesin | CAS_31078-12-3)
Affinity DataKi:  3.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85498(CAS_5486808 | Litorin | NSC_5486808)
Affinity DataKi:  4.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  4.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85496(DPhe6-Bn(6-13)methylester)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85502(PG-L)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85493(DTyr6,DAla11-Bn(6-13)butylamide)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85487(Leu8-phyllolitorin)
Affinity DataKi:  5.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85500(Bombesin,Phe13)
Affinity DataKi:  6.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85499(CAS_29451-71-6 | NSC_5489061 | Ranatensin)
Affinity DataKi:  6.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85478(Bombesin, SAP | CAS_31362-50-2)
Affinity DataKi:  7.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  7.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM81964(CAS_5486814 | Gastrin | NSC_5486814 | Neuromedin C)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85491(Leu13,Psi(CH2NH),Leu14-BN)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85492(GRP-10,frog)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85486(DPhe6-Bn[6-14))
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85485(DPhe6-Bn(6-13)NHN(ME)2)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50071745(CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Trp-Ala-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85479(DPhe6-Bn(1-13)NH2)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85490(DPhe6,Leu13,Psi(CH2NH),Cpa14-Bn(6-14))
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85489(DPhe6,12,Leu14-Bn)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85503(Dphe12-Bn)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 921 total ) | Next | Last >>
Jump to: