Compile Data Set for Download or QSAR
maximum 50k data
Found 2063 Enz. Inhib. hit(s) with Target = 'Casein kinase I isoform delta'
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50105742(4-[4-(4-Fluoro-phenyl)-5-(2-methoxy-pyrimidin-4-yl...)
Affinity DataKi:  25nMAssay Description:Binding affinity to CK1delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKi:  39nMAssay Description:Binding affinity to CK1delta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50537592(CHEMBL4632881)
Affinity DataKi:  40nMAssay Description:Inhibitory activity against HIV-1 Y181C reverse transcriptase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM25116(1-tert-butyl-3-(4-methylphenyl)-1H-pyrazolo[3,4-d]...)
Affinity DataKi:  1.06E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM50142887(1-(tert-butyl)-3-(4-chlorophenyl)-4-aminopyrazolo[...)
Affinity DataKi:  1.29E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50402020(CHEMBL2205426)
Affinity DataKi: >7.80E+3nMAssay Description:Inhibition of recombinant CK1delta after 1 hr by scintillation counter analysis in presence of gamma-[33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM50224883(7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,1...)
Affinity DataKi: >7.83E+3nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM50013720(1-Phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine | C...)
Affinity DataKi:  9.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee

Curated by PDSP Ki Database
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274578(2-fluoro-N-(6-(4-(4- fluorophenyl)-1-(1- (2-hydrox...)
Affinity DataIC50:  0.0340nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274527(N-(6-(4-(4-fluorophenyl)-1- (1-(2-hydroxyethyl)pip...)
Affinity DataIC50:  0.0340nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274525(N-(6-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-imi...)
Affinity DataIC50:  0.0600nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274432(N-(6-(4-(4-fluorophenyl)-1-(piperidin-4-yl)-1H-imi...)
Affinity DataIC50:  0.0640nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274471(N-(6-(1-(1-(2-aminoacetyl)piperidin-4- yl)-4-(4-fl...)
Affinity DataIC50:  0.0850nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274530(N-(6-(1-(1-(2-amino-2- oxoethyl)piperidin-4-yl)-4-...)
Affinity DataIC50:  0.0910nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274618(N-(6-(2-(4-fluorophenyl) imidazo[1,2-a]pyridin-3-y...)
Affinity DataIC50:  0.0960nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM255158(US9475817, 117)
Affinity DataIC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 ul prepared from 15 ul additions of enzyme, substrates (flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM255164(US9475817, 123)
Affinity DataIC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 ul prepared from 15 ul additions of enzyme, substrates (flu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274886(2-Fluoro-N-(6-(2-(4-fluorophenyl)-7-pivaloyl- 5,6,...)
Affinity DataIC50:  0.100nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274453(N-(6-(1-(1-((1,3-dimethyl-1H-pyrazol-4- yl)methyl)...)
Affinity DataIC50:  0.101nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274594(N-(6-(4-(4-fluorophenyl)-1- (2-morpholinoethyl)-1H...)
Affinity DataIC50:  0.104nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274718(N-(6-(4-(4-chlorophenyl)-1-(2- fluoroethyl)-2-meth...)
Affinity DataIC50:  0.109nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274595(N-(6-(4-(4-fluorophenyl)-1- (2-morpholinoethyl)-1H...)
Affinity DataIC50:  0.110nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274713(2-Fluoro-N-(6-(1-(2-fluoroethyl)-4-(4-fluorophenyl...)
Affinity DataIC50:  0.110nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274619(2-(dimethylamino)-N-(6-(2-(4- fluorophenyl)imidazo...)
Affinity DataIC50:  0.111nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274571((S)-2-fluoro-N-(6-(4-(4- fluorophenyl)-2-methyl-1-...)
Affinity DataIC50:  0.112nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274498(N-(6-(1-(1-(3,3- difluorocyclobutanecarbonyl)piper...)
Affinity DataIC50:  0.116nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274720(N-(6-(4-(4-chlorophenyl)-2-methyl- 1-(2,2,2-triflu...)
Affinity DataIC50:  0.126nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274472(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1- (2-hydroxy...)
Affinity DataIC50:  0.128nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274487(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1 isonicotino...)
Affinity DataIC50:  0.130nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274465(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1- (2-methoxy...)
Affinity DataIC50:  0.136nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274513(3,3,3-trifluoropropyl 4-(5-(2-(2- fluoroisonicotin...)
Affinity DataIC50:  0.142nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274500(N-(6-(1-(1-(3- chloropropanoyl)piperidin-4-yl)-4-(...)
Affinity DataIC50:  0.143nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274519(N-(6-(1-(1-(2-amino-2- oxoethyl)piperidin-4-yl)-4-...)
Affinity DataIC50:  0.146nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274690(2-fluoro-N-(6-(4-(4-fluorophenyl)- 1-(2-(1H-pyrazo...)
Affinity DataIC50:  0.147nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274745(6-fluoro-N-(6-(4-(4-fluoro- phenyl)-1,2-dimethyl-1...)
Affinity DataIC50:  0.152nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274544(N-(6-(4-(4-fluorophenyl)-1-(1-(3,3,3-trifluoroprop...)
Affinity DataIC50:  0.159nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274455(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1- ((5-methyl...)
Affinity DataIC50:  0.165nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274704(N-(6-(4-(4-fluorophenyl)-1-(furan-3- ylmethyl)-1H-...)
Affinity DataIC50:  0.169nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274452(N-(6-(1-(1-((1H-pyrazol-5- yl)methyl)piperidin-4-y...)
Affinity DataIC50:  0.170nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274510(US9556179, Compound 80 | oxetan-3-yl 4-(5-(2-(2- f...)
Affinity DataIC50:  0.171nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274501(N-(6-(1-(1-(1- cyanocyclopropanecarbonyl)piperidin...)
Affinity DataIC50:  0.172nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274545(N-(6-(4-(4-fluorophenyl)-1-(1-(isoxazole-3-carbony...)
Affinity DataIC50:  0.173nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274546(N-(6-(4-(4-fluorophenyl)-1- (1-(3,3,3-trifluoropro...)
Affinity DataIC50:  0.175nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274486(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1- (2-hydroxy...)
Affinity DataIC50:  0.178nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274514(US9556179, Compound 84 | methyl 4-(5-(2-(2- fluoro...)
Affinity DataIC50:  0.179nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274454(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1- (2-morphol...)
Affinity DataIC50:  0.183nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274502(N-(6-(1-(1-(1H-imidazole-4- carbonyl)piperidin-4-y...)
Affinity DataIC50:  0.183nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274724(2-fluoro-N-(6-(4-(4-fluoro-3- methylphenyl)-1-(2-f...)
Affinity DataIC50:  0.186nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Christian-Albrechts University Of Kiel

Curated by ChEMBL
LigandPNGBDBM274492(2-fluoro-N-(6-(4-(4-fluorophenyl)-1-(1- (2-morphol...)
Affinity DataIC50:  0.186nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 2063 total ) | Next | Last >>
Jump to: