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Found 26 Enz. Inhib. hit(s) with Target = 'Chymotrypsinogen B2'
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520048(CHEMBL4450993)
Affinity DataKi:  0.420nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520063(CHEMBL4586444)
Affinity DataKi:  0.880nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520058(CHEMBL4469390)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520064(CHEMBL4590739)
Affinity DataKi:  11nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)
Affinity DataKi:  20nMAssay Description:Inhibition of human chymotrypsin by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM247411(US10336754, Example 353 | US11053247, Example 353 ...)
Affinity DataKi:  35nMAssay Description:Binding affinity to human chymotrypsin assessed as inhibition constant using 3-Carbomethoxypropionyl-L-arginyl-Lprolyl-L-tyrosine p-Nitroaniline as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520051(CHEMBL4592765)
Affinity DataKi:  150nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520049(CHEMBL4560112)
Affinity DataKi:  330nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502655(CHEMBL4560512)
Affinity DataKi:  463nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520061(CHEMBL4556207)
Affinity DataKi:  920nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520060(CHEMBL4465306)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520050(CHEMBL4457132)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50504368(CHEMBL4435573)
Affinity DataKi:  1.24E+4nMAssay Description:Inhibition of human chymotrypsin using S-2586 as substrate incubated for 15 mins followed by substrate addition and measured after 1 hr by chromogeni...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50504369(CHEMBL4439549)
Affinity DataKi:  1.63E+4nMAssay Description:Inhibition of human chymotrypsin using S-2586 as substrate incubated for 15 mins followed by substrate addition and measured after 1 hr by chromogeni...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50520052(CHEMBL4554739)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate at pH 8 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50502658(CHEMBL4557877)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533255(CHEMBL4476255)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533255(CHEMBL4476255)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533254(CHEMBL4550207)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533253(CHEMBL4441232)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533253(CHEMBL4441232)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533256(CHEMBL4448473)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533254(CHEMBL4550207)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM513874(bioRxiv20220126.477782, S-217622 | bioRxiv20220126...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human pancreas chymotrypsin using Suc-Ala-Ala-Pro-Phe-AMC as substrate preincubated for 15 mins incubated followed by addition of subst...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50533256(CHEMBL4448473)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human chymotrypsinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B2(Homo sapiens)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50541448(CHEMBL4633785)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of mammalian chymotrypsin (unknown origin) using Suc-AAPF-AMC as substrate preincubated for 10 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed