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Found 7 Enz. Inhib. hit(s) with Target = 'Complement C5'
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50546241(CHEMBL2203296)
Affinity DataIC50:  210nMAssay Description:Inhibition of C5 complement protein in 2% human serum incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50546240(CHEMBL2204196)
Affinity DataIC50:  440nMAssay Description:Inhibition of C5 complement protein in 2% human serum incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50546242(CHEMBL4756677)
Affinity DataIC50:  620nMAssay Description:Inhibition of C5 complement protein in 2% human serum incubated for 15 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50002861(3-(4,5-Diphenyl-oxazol-2-yl)-propionic acid | CHEM...)
Affinity DataKd:  640nMAssay Description:Binding affinity to human C5a assessed as dissociation constant after 1 hr by circular dichroism analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50097346((+/-)-2-(3-chloro-9H-carbazol-7-yl)propanoic acid ...)
Affinity DataKd:  580nMAssay Description:Binding affinity to human C5a assessed as dissociation constant after 1 hr by circular dichroism analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50103504(CHEBI:9352 | Clinoril | Sulindac)
Affinity DataKd:  570nMAssay Description:Binding affinity to human C5a assessed as dissociation constant after 1 hr by circular dichroism analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetComplement C5(Homo sapiens)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)
Affinity DataKd:  710nMAssay Description:Binding affinity to human C5a assessed as dissociation constant after 1 hr by circular dichroism analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed