TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of DCAMKL2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of DCAMKL2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >9.57E+3nMAssay Description:Inhibition of DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 83.5nMAssay Description:Inhibition of human DCAMKL2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 94.4nMAssay Description:Inhibition of human DCAMKL2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of DCAMKL2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human DCAMKL2 using [KKALRRQETVDAL] as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human DCAMKL2 (376 to end residues) using KKLNRTLSFAEPG as substrate after 40 mins in presence of [gamma-33ATP] by radiomet...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DCAMKL2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]LSD from Homo sapiens (human) 5-HT6 receptor expressed in Homo sapiens (human) HEK293 cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 4.50E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 73nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 4.50E+3nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 73nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 73nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase DCLK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DCAMKL2 kinase domainMore data for this Ligand-Target Pair