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Found 2 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase FKBP3'
TargetPeptidyl-prolyl cis-trans isomerase FKBP3(Homo sapiens (Human))
Max Planck Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50263407(CHEMBL4090599)
Affinity DataKi:  1.13E+3nMAssay Description:Displacement of 5-(3-(4-(((5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-5-vinyl-3,10-diazabicyclo[4.3.1]decan-3-yl)methyl)-1H-1,2,3-triazol-1-yl)prop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP3(Homo sapiens (Human))
Max Planck Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM50080528(3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2-oxocyclohexyl)...)
Affinity DataKi:  1.24E+5nMAssay Description:Inhibition constant(Ki) for inhibition of PPIase activity of L. pneumophilia FK506 binding protein 25 (Conc=40 nM) of FKBPsfamilyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed