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Found 40 Enz. Inhib. hit(s) with Target = 'Env polyprotein'
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50333241(CHEMBL254781 | N-(4-chlorophenyl)-N'-(2,2,6,6-tetr...)
Affinity DataIC50:  610nMAssay Description:Inhibition of HIV-1 isolate YTA48P HIV-1 gp120More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023611(CHEMBL2380932)
Affinity DataIC50:  2.84E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023610(CHEMBL3341857)
Affinity DataIC50:  8.31E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023609(CHEMBL3341856)
Affinity DataIC50:  8.31E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023608(CHEMBL3341855)
Affinity DataIC50:  8.31E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023614(CHEMBL3341854)
Affinity DataIC50:  8.31E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023613(CHEMBL3341853)
Affinity DataIC50:  8.31E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023612(CHEMBL3341852)
Affinity DataIC50:  8.31E+3nMAssay Description:Inhibition of HIV1 gp41 NHR assessed as inhibition of 6HB formation by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023609(CHEMBL3341856)
Affinity DataEC50:  3.40nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023608(CHEMBL3341855)
Affinity DataEC50:  7.90nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023614(CHEMBL3341854)
Affinity DataEC50:  3.90nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023613(CHEMBL3341853)
Affinity DataEC50:  44nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50072279(CHEMBL3408356)
Affinity DataKd:  452nMAssay Description:Binding affinity to HIV1 gp41 (46 residues) by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023619(CHEMBL3341851)
Affinity DataEC50:  327nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023620(CHEMBL3341850)
Affinity DataEC50:  197nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023621(CHEMBL3341849)
Affinity DataEC50:  29nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023622(CHEMBL3341848)
Affinity DataEC50:  52nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023623(CHEMBL3341847)
Affinity DataEC50:  15nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023624(CHEMBL3341846)
Affinity DataEC50:  176nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023625(CHEMBL3341845)
Affinity DataEC50:  145nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023626(CHEMBL3341844)
Affinity DataEC50:  89nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023623(CHEMBL3341847)
Affinity DataEC50:  117nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023614(CHEMBL3341854)
Affinity DataEC50:  13nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023615(CHEBI:608828 | DP178 | Enfuvirtide | Fuzeon | Fuze...)
Affinity DataEC50:  14nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023611(CHEMBL2380932)
Affinity DataEC50:  1.30nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023623(CHEMBL3341847)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023614(CHEMBL3341854)
Affinity DataEC50:  139nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023615(CHEBI:608828 | DP178 | Enfuvirtide | Fuzeon | Fuze...)
Affinity DataEC50:  542nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023611(CHEMBL2380932)
Affinity DataEC50: >1.00E+3nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50072278(CHEMBL3408357)
Affinity DataKd:  250nMAssay Description:Binding affinity to HIV1 gp41 (46 residues) by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023615(CHEBI:608828 | DP178 | Enfuvirtide | Fuzeon | Fuze...)
Affinity DataKd:  182nMAssay Description:Binding affinity to HIV1 gp41 (46 residues) by surface plasmon resonance methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023610(CHEMBL3341857)
Affinity DataEC50:  3.30nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM23208((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-17-hydroxy-1,...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50346601(NSC-114945 | OLEANOLIC_ACID | Oleanolic acid | Ole...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023618(CHEMBL3341858)
Affinity DataEC50:  3.24E+3nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023617(CHEMBL3341859)
Affinity DataEC50:  3.58E+3nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023616(CHEMBL3341860)
Affinity DataEC50:  2.18E+3nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023615(CHEBI:608828 | DP178 | Enfuvirtide | Fuzeon | Fuze...)
Affinity DataEC50:  10nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnv polyprotein(Human immunodeficiency virus 1)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50023612(CHEMBL3341852)
Affinity DataEC50:  20nMAssay Description:Inhibition of HIV1 gp41-induced cell-cell fusion between viral envelope expressing human HL2/3 cells to CD4/CCR5 receptor expressing TZM-bl cells aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed