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Found 91 Enz. Inhib. hit(s) with Target = 'Putative sugar transporter'
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216468((3R,4S,5S,6R)-6-(hydroxymethyl)-3-(undec-10-enylox...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179097((3R,4S,5R,6R)-4-(decyloxy)-6-(hydroxymethyl)-tetra...)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179112((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(undecyloxy)-tet...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179102((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(undec-10-enylox...)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179091((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(octyloxy)-tetra...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179111((3R,4S,5R,6R)-4-(dodecyloxy)-6-(hydroxymethyl)-tet...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179094((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(nonyloxy)-tetra...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179093((3R,4S,5R,6R)-4-(dodec-11-enyloxy)-6-(hydroxymethy...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179098((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(pentadec-14-eny...)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179100((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(non-8-enyloxy)-...)
Affinity DataKi:  4.10E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179109((3R,4S,5R,6R)-4-(dec-9-enyloxy)-6-(hydroxymethyl)-...)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179102((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(undec-10-enylox...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179108((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(5-phenylpentylo...)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179099((3R,4S,5R,6R)-4-(5-(4-butylphenyl)pentyloxy)-6-(hy...)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179095((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(8,8,9,9,10,10,1...)
Affinity DataKi:  1.30E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179092((3R,4S,5S,6R)-6-(hydroxymethyl)-4-((Z)-20-((3S,4R,...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179106((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(8-phenyloctylox...)
Affinity DataKi:  1.48E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179110((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(4,4,5,5,6,6,7,7...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179107((3R,4S,5R,6R,E)-4-(hexadec-7-enyloxy)-6-(hydroxyme...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179104((3R,4S,5R,6R)-4-(2-(allyloxy)ethoxy)-6-(hydroxymet...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179105((3R,4S,5R,6R)-4-(7-(allyloxy)heptyloxy)-6-(hydroxy...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179101((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(tetradecyloxy)-...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179096((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(octadecyloxy)-t...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179090(CHEMBL203457 | methyl 16-((3R,4S,5R,6R)-2,3,5-trih...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216470((2R,3R,4R,5S)-2-((R)-1,2-dihydroxyethyl)-5-(undec-...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216471((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(undec-10-eny...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216465((2R,3S,4S,5R,6R)-2-(hydroxymethyl)-6-(undec-10-eny...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216467((2R,3R,4R,5R)-2-((R)-1,2-dihydroxyethyl)-5-(undec-...)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179089((3R,4S,5S,6R)-6-(hydroxymethyl)-4-(20-((3S,4R,5R,6...)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50179103((3R,4S,5R,6R)-6-(hydroxymethyl)-4-(2-(non-8-enylox...)
Affinity DataKi:  5.90E+5nMAssay Description:Inhibition of D-glucose uptake mediated by PfHT expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216466((3R,4R,5S)-5-((R)-2-hydroxy-1-(undec-10-enyloxy)et...)
Affinity DataKi:  1.50E+6nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM50216469((3R,4S,5S,6R)-6-((undec-10-enyloxy)methyl)-tetrahy...)
Affinity DataKi:  2.00E+6nMAssay Description:Inhibition of [3H]glucose uptake at Plasmodium falciparum HT expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453221(US10729691, Example 6)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453222(US10729691, Example 7)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453231(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-1-methy...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453233(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-1-methy...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453242(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-5,7-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453243(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-5,7-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453253(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-6-methy...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453255(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453256(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453258(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)thieno[3...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453259(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-6-acety...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453260(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-6-acety...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453261(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453262(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453263(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-6-acety...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453264(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453265(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPutative sugar transporter(Plasmodium falciparum)
Université

Curated by ChEMBL
LigandPNGBDBM453270(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-6-acety...)
Affinity DataIC50:  55nMAssay Description:Parasite cultures were seeded in 96-well plates (1% hematocrit, 1-2% starting parasitemia, 100 μL total volume) with varying concentrations of t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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